SCHEMBL13197844

SCHEMBL13197844

C[C@H](Cc1ccc(N)cc1)NC(=O)OC(C)(C)C

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.52
RAB9A P51151 2/20 0.52
ATM Q13315 1/20 0.47
CTSS P25774 6/20 0.46
CTSK P43235 5/20 0.46
ACACB O00763 2/20 0.46
CA2 P00918 3/20 0.46
CTSL P07711 1/20 0.45
CTSB P07858 1/20 0.45
KLK5 Q9Y337 1/20 0.44
ITGB3 P05106 1/20 0.44
ITGA2B P08514 1/20 0.44
CA1 P00915 1/20 0.43
CA4 P22748 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
ACE P12821 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6763468 1.00 NPC1 (0.52) NPC1RAB9AATMCTSSCTSK
SCHEMBL8543180 0.87 CTSS (0.60) NPC1RAB9AATMCTSSCTSK
SCHEMBL2742779 0.87 ACACB (0.54) NPC1RAB9AATMCTSSCTSK
SCHEMBL13446081 0.87 CTSS (0.60) NPC1RAB9AATMCTSSCTSK
SCHEMBL14588983 0.87 ACACB (0.54) NPC1RAB9AATMCTSSCTSK
SCHEMBL23279494 0.85 ACACB (0.59) NPC1RAB9AATMCTSSCTSK
SCHEMBL30101873 0.85 CTSS (0.60) NPC1RAB9AATMCTSSCTSK
SCHEMBL165908 0.85 CYP1A2 (0.49) NPC1RAB9AATMCTSSCTSK
SCHEMBL255673 0.85 CTSS (0.60) NPC1RAB9AATMCTSSCTSK
SCHEMBL26703849 0.85 ACACB (0.55) ATMCTSSCTSKACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7776891-B2 VLA-4 antagonists MERCK SHARP & DOHME CORP. (US) 2010-08-17 US disclosed
US-20070219252-A1 Vla-R Antagonists MERCK SHARP & DOHME LLC 2007-09-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070219252-A1 Vla-R Antagonists VCAM1, LTB4R, ITGA4 NPC1 3964/4885RAB9A 1244/4885ATM 4830/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.