SCHEMBL13201540

SCHEMBL13201540

CC(=O)NCc1nccnc1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.40
ALDH1A1 P00352 3/20 0.38
POLB P06746 2/20 0.38
MAPT P10636 2/20 0.38
RAB9A P51151 2/20 0.38
KMT2A Q03164 2/20 0.37
SETDB1 Q15047 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
NPC1 O15118 1/20 0.35
HTT P42858 1/20 0.35
VHL P40337 1/20 0.35
NOTUM Q6P988 1/20 0.35
MALT1 Q9UDY8 1/20 0.35
MAPKAPK2 P49137 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23042833 0.88 L3MBTL1 (0.33) NPSR1L3MBTL1ALDH1A1KMT2ACYP1A2
SCHEMBL29561964 0.82 CYP1A2 (0.38) NPSR1ALDH1A1POLBMAPTRAB9A
SCHEMBL19652463 0.82 CYP1A2 (0.38) NPSR1ALDH1A1POLBMAPTRAB9A
SCHEMBL13218642 0.81 HPGD (0.33) NPSR1ALDH1A1POLBKMT2ACYP1A2
SCHEMBL14617245 0.81 PTGES (0.43) L3MBTL1ALDH1A1MAPTKMT2ACYP1A2
SCHEMBL1128663 0.81 KMT2A (0.32) NPSR1ALDH1A1KMT2ACYP1A2CYP2C9
SCHEMBL29636346 0.81 PTGES (0.43) L3MBTL1ALDH1A1MAPTKMT2ACYP1A2
SCHEMBL12436062 0.81 PTGES (0.40) L3MBTL1ALDH1A1POLBMAPTHDAC6
SCHEMBL31330611 0.80 EGLN1 (0.42) ALDH1A1POLBMAPTRAB9AKMT2A
SCHEMBL31391134 0.80 KDM4E (0.33) NPSR1ALDH1A1KMT2ACYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 40 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122055366-A GCN2 and PERK kinase modulators and methods of use thereof 德西费拉制药有限责任公司 2026-05-15 CN disclosed
EP-4719606-A2 GCN2 AND PERK KINASE MODULATORS AND METHODS OF USE THEREOF Deciphera Pharmaceuticals, LLC (US) 2026-04-08 EP disclosed
US-12180210-B2 Compounds INTRA-CELLULAR THERAPIES, INC. (US) 2024-12-31 US disclosed
US-12162890-B2 Heteroaromatic NMDA receptor modulators and uses thereof NOVARTIS AG (CH) 2024-12-10 US disclosed
WO-2024249493-A2 GCN2 AND PERK KINASE MODULATORS AND METHODS OF USE THEREOF DECIPHERA PHARMACEUTICALS, LLC (US) 2024-12-05 WO disclosed
EP-3870300-B1 IMIDAZO[1,5-A]PYRAZINE COMPOUNDS AS PDE2 INHIBITORS INTRA CELLULAR THERAPIES INC (US) 2024-07-10 EP disclosed
US-20230192691-A1 HETEROCYCLIC COMPOUNDS AS BTK INHIBITORS BEIJING INNOCARE PHARMA TECH CO LTD (CN) 2023-06-22 US disclosed
US-20230023543-A1 HETEROAROMATIC NMDA RECEPTOR MODULATORS AND USES THEREOF NOVARTIS AG (CH) 2023-01-26 US disclosed
US-20230023543-A1 HETEROAROMATIC NMDA RECEPTOR MODULATORS AND USES THEREOF NOVARTIS AG (CH) 2023-01-26 US disclosed
CN-110627796-B Nitrogenous heterocyclic derivative and application thereof in medicine 北京越之康泰生物医药科技有限公司 2022-07-12 CN disclosed
WO-2016106106-A2 FUSED HETEROARYL DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-06-30 WO disclosed
WO-2016106106-A2 FUSED HETEROARYL DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-06-30 WO disclosed
US-20140221333-A1 BTK INHIBITORS MERCK SHARP & DOHME B.V. (NL) 2014-08-07 US disclosed
CN-103917545-A BTK inhibitors MERCK SHARP & DOHME 2014-07-09 CN disclosed
EP-2734529-A1 BTK INHIBITORS Merck Sharp & Dohme Corp. (US) 2014-05-28 EP disclosed
WO-2013010380-A1 BTK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2013-01-24 WO disclosed
EP-2548877-A1 4-(5-Membered fused pyridinyl)benzamides as BTK-inhibitors MSD Oss B.V. (NL) 2013-01-23 EP disclosed
EP-2548877-A1 4-(5-Membered fused pyridinyl)benzamides as BTK-inhibitors MSD Oss B.V. (NL) 2013-01-23 EP disclosed
US-7772231-B2 Substituted pyrazolo[3,4-d]pyrimidines as protein kinase inhibitors ABBOTT LABORATORIES (US) 2010-08-10 US disclosed
US-20070203143-A1 PROTEIN KINASE INHIBITORS ABBVIE INC. 2007-08-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12162890-B2 Heteroaromatic NMDA receptor modulators and uses thereof GRIN2C, GRIN2A, GRIN1 NPSR1 61/4885L3MBTL1 4411/4885ALDH1A1 1771/4885
US-20230192691-A1 HETEROCYCLIC COMPOUNDS AS BTK INHIBITORS BTK, SYK, LYN NPSR1 3733/4885L3MBTL1 872/4885ALDH1A1 3975/4885
US-20230023543-A1 HETEROAROMATIC NMDA RECEPTOR MODULATORS AND USES THEREOF GRIN2C, GRIN2A, GRIN1 NPSR1 61/4885L3MBTL1 4411/4885ALDH1A1 1771/4885
US-12180210-B2 Compounds PDE2A, PDE3A, PDE3B NPSR1 1682/4885L3MBTL1 4784/4885ALDH1A1 519/4885
US-20140221333-A1 BTK INHIBITORS BTK, SYK, ABL1 NPSR1 4712/4885L3MBTL1 2121/4885ALDH1A1 4482/4885
US-20070203143-A1 PROTEIN KINASE INHIBITORS PACSIN2, MAP3K20, PHKG1 NPSR1 4339/4885L3MBTL1 1942/4885ALDH1A1 4453/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.