SCHEMBL13209596

SCHEMBL13209596

O=C1C=CC2(CCNCC2)N1c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 4/20 0.45
TSHR P16473 5/20 0.45
USP2 O75604 6/20 0.44
CYP2D6 P10635 6/20 0.44
ALDH1A1 P00352 5/20 0.40
CYP3A4 P08684 4/20 0.40
CYP2C19 P33261 2/20 0.40
MMP13 P45452 1/20 0.40
SIGMAR1 Q99720 3/20 0.39
OPRM1 P35372 1/20 0.39
HTR3E A5X5Y0 1/20 0.39
HTR3B O95264 1/20 0.39
ADRB1 P08588 1/20 0.39
HTR3A P46098 1/20 0.39
HTR3D Q70Z44 1/20 0.39
HTR3C Q8WXA8 1/20 0.39
CYP1A2 P05177 4/20 0.38
TP53 P04637 3/20 0.38
MAPK1 P28482 3/20 0.38
HIF1A Q16665 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14232651 0.84 MGLL (0.35) HSD17B10TSHRUSP2CYP2D6ALDH1A1
SCHEMBL2990811 0.79 MEN1 (0.51) HSD17B10TSHRCYP2D6ALDH1A1CYP3A4
SCHEMBL8811652 0.71 HSD17B10 (0.58) HSD17B10TSHRUSP2CYP2D6ALDH1A1
SCHEMBL7883556 0.71 HSD17B10 (0.46) HSD17B10TSHRUSP2CYP2D6ALDH1A1
SCHEMBL14209241 0.70 MMP13 (0.54) HSD17B10TSHRUSP2CYP2D6ALDH1A1
Hydrochloric Acid SCHEMBL7883554 0.70 HSD17B10 (0.45) HSD17B10TSHRUSP2CYP2D6ALDH1A1
SCHEMBL14834366 0.70 OPRM1 (0.38) ALDH1A1OPRM1HTR2CHTR2B
SCHEMBL20764919 0.69 GSK3A (0.31) HSD17B10OPRM1MGLL
Hydrochloric Acid SCHEMBL2990834 0.69 MMP13 (0.53) HSD17B10TSHRUSP2CYP2D6ALDH1A1
SCHEMBL17149455 0.68 TSHR (0.46) HSD17B10TSHRUSP2CYP2D6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7786308-B2 Muscarinic modulators VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-08-31 US disclosed
US-7786308-B2 Muscarinic modulators VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-08-31 US disclosed