SCHEMBL13239488

SCHEMBL13239488

COC(=O)[C@H](Cc1ccc(N(C(C)=O)C(C)=O)cc1)N(C)P

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.38
ESR2 Q92731 1/20 0.38
PTPRB P23467 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.36
ALDH1A1 P00352 2/20 0.36
NPC1 O15118 2/20 0.36
KDM4E B2RXH2 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
HSD17B10 Q99714 1/20 0.36
ACACB O00763 1/20 0.36
POLB P06746 1/20 0.35
PPARG P37231 3/20 0.34
PPARD Q03181 3/20 0.34
PPARA Q07869 3/20 0.34
CRHBP P24387 1/20 0.34
CRHR2 Q13324 1/20 0.34
MIF P14174 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12904040 0.91 ESR1 (0.37) ESR1ESR2PTPRBSMN1; SMN2ALDH1A1
SCHEMBL12904053 0.89 PTPRB (0.33) ESR1ESR2PTPRBSMN1; SMN2ALDH1A1
SCHEMBL13239494 0.85 SMN1; SMN2 (0.40) ESR1ESR2PTPRBSMN1; SMN2ALDH1A1
SCHEMBL10329642 0.82 ESR1 (0.34) ESR1ESR2PTPRBSMN1; SMN2ALDH1A1
SCHEMBL10329633 0.81 ESR1 (0.41) ESR1ESR2PTPRBNPC1PPARG
SCHEMBL12904046 0.81 MEN1 (0.51) PTPRBSMN1; SMN2KDM4ETSHRMAPK1
SCHEMBL13239493 0.80 PTPRB (0.46) ESR1ESR2PTPRBALDH1A1PPARG
SCHEMBL12904067 0.77 PTPRB (0.39) ESR1ESR2PTPRBSMN1; SMN2ALDH1A1
SCHEMBL12904044 0.76 SAE1 (0.43) ESR1ESR2PTPRBSMN1; SMN2ALDH1A1
SCHEMBL12904068 0.76 PTPRB (0.54) PTPRBSMN1; SMN2ALDH1A1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7759388-B2 Phenylalanine derivatives AJINOMOTO CO., INC. (JP) 2010-07-20 US disclosed
US-20090048236-A1 NEW PHENYLALANINE DERIVATIVES AJINOMOTO CO. INC (JP) 2009-02-19 US disclosed
US-7452905-B2 Phenylalanine derivatives AJINOMOTO CO., INC. (JP) 2008-11-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090048236-A1 NEW PHENYLALANINE DERIVATIVES ITGB4, VCAM1, ITGA4 ESR1 2563/4885ESR2 2887/4885PTPRB 513/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.