SCHEMBL13245993

SCHEMBL13245993

Cc1ccc(-c2ccc(S(=O)(=O)Nc3cccc(NC(=O)C(C)(C)N)c3)cc2F)o1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.48
GHSR Q92847 12/20 0.46
L3MBTL1 Q9Y468 1/20 0.40
IDH2 P48735 2/20 0.40
PIK3CD O00329 1/20 0.39
PIK3CA P42336 1/20 0.39
PIK3CB P42338 1/20 0.39
PIK3CG P48736 1/20 0.39
PRKDC P78527 1/20 0.39
PIK3C3 Q8NEB9 1/20 0.39
PKM P14618 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4664054 0.91 KDM4E (0.45) KDM4EGHSRPIK3CDPIK3CAPIK3CB
SCHEMBL2997886 0.89 KDM4E (0.47) KDM4EGHSRL3MBTL1IDH2
SCHEMBL13245995 0.88 GHSR (0.47) KDM4EGHSRIDH2
SCHEMBL4664052 0.85 HTT (0.47) GHSRPIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL4664203 0.85 GHSR (0.44) KDM4EGHSRPKM
SCHEMBL13245951 0.84 ALDH1A1 (0.46) KDM4EGHSRL3MBTL1
SCHEMBL2984221 0.82 HTR6 (0.52) KDM4EGHSRL3MBTL1PKM
SCHEMBL4793678 0.80 GHSR (0.46) KDM4EGHSRPIK3CDPIK3CAPIK3CB
SCHEMBL2984133 0.77 GHSR (0.43) KDM4EGHSRL3MBTL1PIK3CDPIK3CA
SCHEMBL2989098 0.77 GHSR (0.49) GHSRL3MBTL1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100179168-A1 ARYL AND HETEROARYL SULPHONAMIDES AS GROWTH HORMONE SECRETAGOGUE RECEPTOR AGONISTS BLANEY EMMA LOUISE 2010-07-15 US disclosed
US-20100179168-A1 ARYL AND HETEROARYL SULPHONAMIDES AS GROWTH HORMONE SECRETAGOGUE RECEPTOR AGONISTS BLANEY EMMA LOUISE 2010-07-15 US disclosed
WO-2007118852-A1 ARYL AND HETEROARYL SULPHONAMIDES AS GROWTH HORMONE SECRETAGOGUE RECEPTOR AGONISTS GLAXO GROUP LIMITED (GB) 2007-10-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100179168-A1 ARYL AND HETEROARYL SULPHONAMIDES AS GROWTH HORMONE SECRETAGOGUE RECEPTOR AGONISTS GHSR, GHRHR, GIPR KDM4E 3009/4885GHSR 1/4885L3MBTL1 4612/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.