SCHEMBL132547

SCHEMBL132547

[CH]1Cc2ccccc2CO1

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.34
MAOB P27338 2/20 0.34
TSHR P16473 1/20 0.33
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CYP1A2 P05177 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14591142 0.75 MAOA (0.32) MAOAMAOBTSHRCA1CA2
SCHEMBL8535446 0.75 MAOA (0.39) MAOAMAOBTSHRCA1CA2
SCHEMBL25345416 0.69 TRPA1 (0.33)
SCHEMBL29471383 0.67
SCHEMBL59871 0.67
SCHEMBL30473446 0.67 TSHR (0.42) MAOAMAOBTSHRCA1CA2
SCHEMBL4486486 0.67 TSHR (0.42) MAOAMAOBTSHRCA1CA2
SCHEMBL19348293 0.67 OXTR (0.41) MAOAMAOBTSHRNPC1RAB9A
Ammonia Solution, Strong SCHEMBL23320033 0.65 MAOA (0.40) MAOAMAOBTSHRCA1CA2
SCHEMBL16439994 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 155 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023148206-A1 MICROBIOCIDAL N-AMIDE DERIVATIVES SYNGENTA CROP PROTECTION AG (CH) 2023-08-10 WO claimed
EP-2134342-B1 MONOCYCLIC ANILIDE SPIROLACTAM CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME (US) 2013-01-30 EP claimed
CN-117642185-A Improved CD30 targeting antibody drug conjugates and uses thereof 路德维希-马克西米利安慕尼黑大学 2024-03-01 CN disclosed
WO-2024010015-A1 PYRIMIDINE DERIVATIVES あすか製薬株式会社 2024-01-11 WO disclosed
WO-2023148206-A1 MICROBIOCIDAL N-AMIDE DERIVATIVES SYNGENTA CROP PROTECTION AG (CH) 2023-08-10 WO disclosed
US-11542261-B2 Substituted Imidazo[1,2-a]-pyridines as IRAK 1/4 and FLT3 inhibitors CHILDREN'S HOSPITAL MEDICAL CENTER (US) 2023-01-03 US disclosed
US-20220213094-A1 Substituted Imidazo[l,2-a]-pyridines as IRAK 1/4 and FLT3 Inhibitors CHILDREN'S HOSPITAL MEDICAL CENTER (US) 2022-07-07 US disclosed
CN-108137513-B Pyrimidine derivatives ASKA 制药株式会社 2022-03-01 CN disclosed
US-11254667-B2 Substituted imidazo[1,2-A]pyridines as IRAK 1/4 and flt3 inhibitors CHILDREN'S HOSPITAL MEDICAL CENTER (US) 2022-02-22 US disclosed
US-11160785-B2 Methods and compositions for improving cognitive function AGENEBIO INC. (US) 2021-11-02 US disclosed
EP-3372589-B1 PYRIMIDINE DERIVATIVE ASKA PHARM CO LTD (JP) 2021-10-20 EP disclosed
EP-0627400-A1 Aromatic acetylcholinesterase inhibitors MERRELL DOW PHARMACEUTICALS INC. (US) 1994-12-07 EP disclosed
EP-0612729-A2 Pyridine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1994-08-31 EP disclosed
EP-0611769-A1 Silylated acetylcholinesterase inhibitors MERRELL DOW PHARMACEUTICALS INC. (US) 1994-08-24 EP disclosed
EP-0291787-B1 Novel substituted silyl alkylene amines MERRELL DOW PHARMA (US) 1994-03-16 EP disclosed
US-5246948-A Antiinflammatory, antipyretic, analgesic, antiallergic, immunosupressing or immunomodulating activity TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-09-21 US disclosed
EP-0522606-A2 Pyridine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-01-13 EP disclosed
EP-0409676-A1 Novel acetylcholinesterase inhibitors MERRELL DOW PHARMACEUTICALS INC. (US) 1991-01-23 EP disclosed
EP-0403713-A1 Novel acetylcholinesterase inhibitors MERRELL DOW PHARMACEUTICALS INC. (US) 1990-12-27 EP disclosed
EP-0291787-A1 Novel substituted silyl alkylene amines MERRELL DOW PHARMACEUTICALS INC. (US) 1988-11-23 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11254667-B2 Substituted imidazo[1,2-A]pyridines as IRAK 1/4 and flt3 inhibitors IRAK1, IRAK4, FLT3 MAOA 2475/4885MAOB 2677/4885TSHR 2789/4885
US-11160785-B2 Methods and compositions for improving cognitive function BACE2, BACE1, GRIN2A MAOA 123/4885MAOB 178/4885TSHR 1591/4885
US-20220213094-A1 Substituted Imidazo[l,2-a]-pyridines as IRAK 1/4 and FLT3 Inhibitors IRAK1, IRAK4, FLT3 MAOA 2515/4885MAOB 2629/4885TSHR 2908/4885
US-11542261-B2 Substituted Imidazo[1,2-a]-pyridines as IRAK 1/4 and FLT3 inhibitors IRAK1, IRAK4, IRAK2 MAOA 3606/4885MAOB 3580/4885TSHR 2194/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.