SCHEMBL13268696

SCHEMBL13268696

COc1cc(Cn2cnc3c(N)ncnc32)ccc1O

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 8/20 0.56
PI4KA P42356 3/20 0.56
PI4K2B Q8TCG2 3/20 0.56
PI4K2A Q9BTU6 3/20 0.56
PI4KB Q9UBF8 3/20 0.56
NSD3 Q9BZ95 1/20 0.50
ADORA1 P30542 4/20 0.49
MEN1 O00255 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2C9 P11712 1/20 0.47
KMT2A Q03164 1/20 0.47
ADORA2B P29275 1/20 0.47
AHCY P23526 2/20 0.46
LMNA P02545 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
HPGD P15428 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11862441 0.89 ADORA2A (0.60) ADORA2API4KAPI4K2BPI4K2API4KB
SCHEMBL3395858 0.83 HSP90AA1 (0.62) ADORA2API4KAPI4K2BPI4K2API4KB
SCHEMBL1422156 0.80 NSD3 (0.70) ADORA2API4KAPI4K2BPI4K2API4KB
SCHEMBL11811272 0.78 ADORA2A (0.64) ADORA2API4KAPI4K2BPI4K2API4KB
SCHEMBL6381371 0.77 ADORA2A (0.63) ADORA2API4KAPI4K2BPI4K2API4KB
SCHEMBL288237 0.77 ADORA2A (0.71) ADORA2API4KAPI4K2BPI4K2API4KB
SCHEMBL11827194 0.75 HDAC6 (0.54) HPGD
SCHEMBL21788552 0.74 ADORA2A (0.76) ADORA2API4KAPI4K2BPI4K2API4KB
SCHEMBL6659204 0.73 ADORA2A (0.74) ADORA2API4KAPI4K2BPI4K2API4KB
9-Benzyl-9H-Adenine SCHEMBL104932 0.73 ADORA2A (1.00) ADORA2API4KAPI4K2BPI4K2API4KB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10174033-B2 N6-substituted adenosine derivatives and N6-substituted adenine derivatives and uses thereof INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 2019-01-08 US disclosed
US-20130045942-A1 N6-SUBSTITUTED ADENOSINE DERIVATIVES AND N6-SUBSTITUTED ADENINE DERIVATIVES AND USES THEREOF INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 2013-02-21 US disclosed
EP-2511283-A1 N6-SUBSTITUTED ADENOSINE DERIVATIVES, N6-SUBSTITUTED ADENINE DERIVATIVES AND USES THEREOF INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 2012-10-17 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10174033-B2 N6-substituted adenosine derivatives and N6-substituted adenine derivatives and uses thereof ADORA2A, ADORA3, ADORA1 ADORA2A 1/4885PI4KA 847/4885PI4K2B 1111/4885
US-20130045942-A1 N6-SUBSTITUTED ADENOSINE DERIVATIVES AND N6-SUBSTITUTED ADENINE DERIVATIVES AND USES THEREOF ADORA2A, ADORA3, ADORA1 ADORA2A 1/4885PI4KA 847/4885PI4K2B 1111/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.