SCHEMBL13282009

SCHEMBL13282009

CCN(c1ccc(OC(F)(F)F)cc1)C1CCN(c2ccc(O)cc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 14/20 0.46
GPR119 Q8TDV5 1/20 0.41
KCNH2 Q12809 1/20 0.40
FFAR4 Q5NUL3 1/20 0.39
CHRM2 P08172 2/20 0.38
HTR2A P28223 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13279655 0.86 CYP3A4 (0.51)
SCHEMBL2098815 0.85 CHRM4 (0.47) CHRM4GPR119KCNH2FFAR4CHRM2
SCHEMBL13281631 0.85 CHRM4 (0.47) CHRM4GPR119KCNH2FFAR4CHRM2
SCHEMBL2056115 0.82 HTR2A (0.55) GPR119KCNH2CHRM2HTR2A
SCHEMBL13279486 0.81 ME2 (0.43) KCNH2
SCHEMBL27474246 0.80 ME3 (0.46) KCNH2CHRM2
SCHEMBL2091318 0.80 CHRM4 (0.53) CHRM4KCNH2CHRM2
SCHEMBL13278861 0.79 CHRM4 (0.59) CHRM4CHRM2
SCHEMBL5536931 0.77 KCNA5 (0.53) CHRM4KCNH2FFAR4
SCHEMBL13281236 0.75 CHRM4 (0.49) CHRM4FFAR4CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2697232-B1 6,7-DIHYDROIMIDAZO[2,1-B][1,3]OXAZINE BACTERICIDES OTSUKA PHARMA CO LTD (JP) 2016-05-18 EP disclosed
US-9051333-B2 6,7-dihydroimidazo [2,1-b] [1,3]oxazine bactericides OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2015-06-09 US disclosed
EP-2697232-A1 6,7 - DIHYDROIMIDAZO [2, 1 - B][1, 3]OXAZINE BACTERICIDES OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2014-02-19 EP disclosed
US-20140031342-A1 6,7-DIHYDROIMIDAZO [2,1-b] [1,3]OXAZINE BACTERICIDES OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2014-01-30 US disclosed
WO-2012141338-A1 6,7 - DIHYDROIMIDAZO [2, 1 - B] [1, 3] OXAZINE BACTERICIDES OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2012-10-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140031342-A1 6,7-DIHYDROIMIDAZO [2,1-b] [1,3]OXAZINE BACTERICIDES BRD1, OXA1L, QDPR CHRM4 1329/4885GPR119 2371/4885KCNH2 600/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.