SCHEMBL13316614

SCHEMBL13316614

Fc1ccc(Cc2cccc(Cl)c2F)cn1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42
MPO P05164 1/20 0.39
P2RX7 Q99572 3/20 0.36
CYP11B2 P19099 2/20 0.36
CYP11B1 P15538 1/20 0.36
AKR1B1 P15121 1/20 0.35
GRIN1 Q05586 2/20 0.34
GRIN2B Q13224 2/20 0.34
SGMS2 Q8NHU3 1/20 0.33
RXRA P19793 1/20 0.33
CNR2 P34972 1/20 0.32
PNMT P11086 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13316625 0.83 MPO (0.41) MPOP2RX7AKR1B1GRIN1GRIN2B
SCHEMBL13316638 0.79 MPO (0.34) MPOAKR1B1GRIN1GRIN2BRXRA
SCHEMBL13316629 0.75 MPO (0.36) MPOAKR1B1GRIN1GRIN2BSGMS2
SCHEMBL13316673 0.73 PDE10A (0.39) MPO
SCHEMBL13349598 0.72 CXCR2 (0.32) MPOGRIN1GRIN2BRXRACNR2
SCHEMBL13349597 0.71 CXCR2 (0.34) MPOGRIN1GRIN2BRXRACNR2
SCHEMBL13349673 0.71 MPO (0.32) MPO
SCHEMBL502199 0.70
SCHEMBL29622066 0.70
Hydrochloric Acid SCHEMBL2308988 0.69 CYP11B1 (0.44) CYP11B2CYP11B1GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7745459-B2 Quinolizinone compound and use thereof as HIV integrase inhibitor JAPAN TOBACCO INC. (JP) 2010-06-29 US disclosed
US-7745459-B2 Quinolizinone compound and use thereof as HIV integrase inhibitor JAPAN TOBACCO INC. (JP) 2010-06-29 US disclosed