SCHEMBL13316629

SCHEMBL13316629

N#CCc1ncc(Cc2cccc(Cl)c2F)cn1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MPO P05164 1/20 0.36
AKR1B1 P15121 1/20 0.32
TP53 P04637 1/20 0.32
MDM2 Q00987 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
KMT2A Q03164 1/20 0.32
GRIA1 P42261 1/20 0.32
CACNG8 Q8WXS5 1/20 0.32
SGMS2 Q8NHU3 1/20 0.31
RXRA P19793 1/20 0.30
GRIN1 Q05586 1/20 0.30
GRIN2B Q13224 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13316638 0.84 MPO (0.34) MPOAKR1B1TP53MDM2KDM4E
SCHEMBL13316625 0.81 MPO (0.41) MPOAKR1B1KMT2ASGMS2RXRA
SCHEMBL2744577 0.77 GRIA1 (0.42) MPOAKR1B1MEN1ALDH1A1KMT2A
SCHEMBL13316614 0.75 CYP3A4 (0.42) MPOAKR1B1SGMS2RXRAGRIN1
SCHEMBL13349673 0.74 MPO (0.32) MPOKDM4EMEN1ALDH1A1KMT2A
SCHEMBL21224318 0.69 MEN1 (0.34) MEN1KMT2A
SCHEMBL13316673 0.68 PDE10A (0.39) MPOKDM4EMEN1ALDH1A1KMT2A
SCHEMBL3678639 0.67 MEN1 (0.35) KDM4EMEN1KMT2A
SCHEMBL14252395 0.64 AKR1B1 (0.38) MPOAKR1B1MEN1ALDH1A1KMT2A
SCHEMBL8067746 0.64 ENPP2 (0.44) KDM4EMEN1ALDH1A1KMT2AGRIA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7745459-B2 Quinolizinone compound and use thereof as HIV integrase inhibitor JAPAN TOBACCO INC. (JP) 2010-06-29 US disclosed
US-7745459-B2 Quinolizinone compound and use thereof as HIV integrase inhibitor JAPAN TOBACCO INC. (JP) 2010-06-29 US disclosed