SCHEMBL13345006

SCHEMBL13345006

COC(=O)c1ccc2ccc3c(c2c1)C(CCl)CC3

nearest known ligand 0.53

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 17/20 0.53
MTNR1A P48039 17/20 0.53
MTNR1B P49286 17/20 0.53
LCK P06239 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13345003 0.79 HPGD (0.43) MEN1KMT2A
SCHEMBL3559992 0.72 ADH1A (0.37) LCK
SCHEMBL13131610 0.70 MTNR1A (0.48) MTNR1AMTNR1B
SCHEMBL2259224 0.68 ALDH1A1 (0.44) MTNR1A
SCHEMBL10064018 0.68 LCK (0.41) LCKMEN1KMT2A
SCHEMBL10030448 0.68 LCK (0.41) LCKMEN1KMT2A
SCHEMBL12365494 0.67 ALDH1A1 (0.43) MTNR1AMTNR1B
SCHEMBL785024 0.66 CA12 (0.45) MTNR1AMEN1KMT2A
SCHEMBL16502580 0.66 PDK2 (0.47) MTNR1AMTNR1BLCKMEN1KMT2A
SCHEMBL9644030 0.66 CA1 (0.55) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7718688-B2 Nitrobenzindoles and their use in cancer therapy AUCKLAND UNISERVICES LIMITED (NZ) 2010-05-18 US disclosed
US-20080119442-A1 as hypoxia-selective drugs and radiosensitizers for cancer therapy; nitroreductase inhibitor; 1-(Chloromethyl)-5,6-dinitro-3-(5,6,7-trimethoxyindol-2-carbonyl)-1,2-dihydro-3H-benzo[e]indole; halogenation of naphthalene derivative followed by hydration and cyclization AUCKLAND UNISERVICES LIMITED (NZ) 2008-05-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080119442-A1 as hypoxia-selective drugs and radiosensitizers for cancer therapy; nitroreductase inhibitor; 1-(Chloromethyl)-5,6-dinitro-3-(5,6,7-trimethoxyindol-2-carbonyl)-1,2-dihydro-3H-benzo[e]indole; halogenation of naphthalene derivative followed by hydration and cyclization HIF1AN, HYOU1, HIF1A HTR2C 1207/4885MTNR1A 253/4885MTNR1B 371/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.