SCHEMBL1335633

SCHEMBL1335633

CCCCOc1cccc(-c2c(F)c(F)c(NC(=O)c3ccccc3C(=O)O)c(F)c2F)c1

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 12/20 0.55
NR1H4 Q96RI1 2/20 0.50
NR4A2 P43354 1/20 0.48
AKR1C2 P52895 1/20 0.46
AKR1C1 Q04828 1/20 0.46
PTPN11 Q06124 2/20 0.46
PLK1 P53350 1/20 0.45
THRB P10828 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1335438 0.87 DHODH (0.66) DHODHNR1H4NR4A2AKR1C2AKR1C1
SCHEMBL1337784 0.86 NR1H4 (0.55) DHODHNR1H4NR4A2AKR1C2AKR1C1
SCHEMBL2595923 0.83 DHODH (0.52) DHODHNR1H4NR4A2AKR1C2AKR1C1
SCHEMBL29709148 0.82 DHODH (0.58) DHODHNR1H4NR4A2AKR1C2AKR1C1
SCHEMBL12129672 0.82 DHODH (0.58) DHODHNR1H4NR4A2AKR1C2AKR1C1
SCHEMBL1337478 0.82 DHODH (0.71) DHODHNR1H4NR4A2AKR1C2AKR1C1
SCHEMBL1337021 0.81 DHODH (0.67) DHODHNR4A2
SCHEMBL1335695 0.81 NR1H4 (0.62) DHODHNR1H4NR4A2AKR1C2AKR1C1
SCHEMBL1337732 0.80 NR1H4 (0.56) DHODHNR1H4NR4A2PTPN11THRB
SCHEMBL15928715 0.79 ALDH1A1 (0.58) DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2566847-B1 NOVEL IMMUNOMODULATOR AND ANTI INFLAMMATORY COMPOUNDS ICOZEN THERAPEUTICS PVT LTD (IN) 2018-11-07 EP claimed
US-9758474-B2 Immunomodulator and anti-inflammatory compounds INCOZEN THERAPEUTICS PVT. LTD. (IN) 2017-09-12 US claimed
US-20140220050-A1 NOVEL IMMUNOMODULATOR AND ANTI-INFLAMMATORY COMPOUNDS INCOZEN THERAPEUTICS PVT. LTD. (CH) 2014-08-07 US claimed
US-20110275603-A1 NOVEL IMMUNOMODULATOR AND ANTI-INFLAMMATORY COMPOUNDS RHIZEN PHARMACEUTICALS SA (FR) 2011-11-10 US claimed
EP-2566847-B1 NOVEL IMMUNOMODULATOR AND ANTI INFLAMMATORY COMPOUNDS ICOZEN THERAPEUTICS PVT LTD (IN) 2018-11-07 EP disclosed
US-9758474-B2 Immunomodulator and anti-inflammatory compounds INCOZEN THERAPEUTICS PVT. LTD. (IN) 2017-09-12 US disclosed
US-9758474-B2 Immunomodulator and anti-inflammatory compounds INCOZEN THERAPEUTICS PVT. LTD. (IN) 2017-09-12 US disclosed
US-20140220050-A1 NOVEL IMMUNOMODULATOR AND ANTI-INFLAMMATORY COMPOUNDS INCOZEN THERAPEUTICS PVT. LTD. (CH) 2014-08-07 US disclosed
US-20110275603-A1 NOVEL IMMUNOMODULATOR AND ANTI-INFLAMMATORY COMPOUNDS RHIZEN PHARMACEUTICALS SA (FR) 2011-11-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140220050-A1 NOVEL IMMUNOMODULATOR AND ANTI-INFLAMMATORY COMPOUNDS DHODH, DLD, DHFR DHODH 1/4885NR1H4 1217/4885NR4A2 1697/4885
US-20110275603-A1 NOVEL IMMUNOMODULATOR AND ANTI-INFLAMMATORY COMPOUNDS DHODH, DLD, DHFR DHODH 1/4885NR1H4 1217/4885NR4A2 1697/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.