Lomefloxacin

Lomefloxacin

SCHEMBL133835

CCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CCN[C@@H](C)C3)c(F)c21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

gyrAgyrB

The experimentally established mechanism targets of Lomefloxacin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 1.00
HSD17B10 Q99714 5/20 1.00
ALDH1A1 P00352 5/20 1.00
HPGD P15428 5/20 1.00
PMP22 Q01453 1/20 0.98
KCNH2 Q12809 4/20 0.62
POLB P06746 1/20 0.62
PRKD3 O94806 1/20 0.62
ALOX15 P16050 1/20 0.62
OPRM1 P35372 1/20 0.62
CLK2 P49760 1/20 0.62
CLK4 Q9HAZ1 1/20 0.62
TDP1 Q9NUW8 1/20 0.62
LMNA P02545 3/20 0.54
BRD4 O60885 1/20 0.54
TSHR P16473 1/20 0.54
HTT P42858 1/20 0.54
CYP2J2 P51589 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54
CYP2C9 P11712 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Lomefloxacin SCHEMBL34610 1.00 KDM4E (1.00) KDM4EHSD17B10ALDH1A1HPGDPMP22
Lomefloxacin SCHEMBL29895425 1.00 KDM4E (1.00) KDM4EHSD17B10ALDH1A1HPGDPMP22
Lomefloxacin SCHEMBL34609 1.00 KDM4E (1.00) KDM4EHSD17B10ALDH1A1HPGDPMP22
Lomefloxacin SCHEMBL9226104 1.00 KDM4E (1.00) KDM4EHSD17B10ALDH1A1HPGDPMP22
Lomefloxacin SCHEMBL29388501 1.00 KDM4E (1.00) KDM4EHSD17B10ALDH1A1HPGDPMP22
Lomefloxacin SCHEMBL8912235 0.99 KDM4E (1.00) KDM4EHSD17B10ALDH1A1HPGDPMP22
Lomefloxacin SCHEMBL30034879 0.99 KDM4E (1.00) KDM4EHSD17B10ALDH1A1HPGDPMP22
Lomefloxacin SCHEMBL42051 0.99 KDM4E (1.00) KDM4EHSD17B10ALDH1A1HPGDPMP22
Lomefloxacin SCHEMBL42052 0.99 KDM4E (1.00) KDM4EHSD17B10ALDH1A1HPGDPMP22
Lomefloxacin SCHEMBL2636428 0.99 KDM4E (1.00) KDM4EHSD17B10ALDH1A1HPGDPMP22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1122 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4434588-B1 AEROSOL DELIVERY DEVICE PARI PHARMA GMBH (DE) 2026-04-08 EP claimed
US-20260027140-A1 COMPOSITIONS AND METHODS FOR TREATING AND AMELIORATING RESPIRATORY CONDITIONS AND INFLAMMATION OF MUCOSA ATOPIC MEDICAL INC (US) 2026-01-29 US claimed
EP-3711797-B1 AEROSOL DELIVERY DEVICE PARI PHARMA GMBH (DE) 2025-02-12 EP claimed
EP-3508501-B1 USE OF ANTI-CGRP ANTIBODIES AND ANTIBODY FRAGMENTS TO PREVENT OR INHIBIT PHOTOPHOBIA OR LIGHT AVERSION IN SUBJECTS IN NEED THEREOF, ESPECIALLY MIGRAINE SUFFERERS H LUNDBECK AS (DK) 2024-11-06 EP claimed
EP-4434588-A2 AEROSOL DELIVERY DEVICE AND METHOD OF OPERATING THE AEROSOL DELIVERY DEVICE PARI Pharma GmbH (DE) 2024-09-25 EP claimed
EP-3756665-B1 INTERVAL THERAPY FOR THE TREATMENT OF EYE DISEASES UNIV RAMOT (IL) 2024-08-14 EP claimed
EP-3374391-B1 ANTIBODY MOLECULE-DRUG CONJUGATES THAT SPECIFICALLY BINDS TO LIPOPOLYSACCHARIDE AND USES THEREOF VISTERRA INC (US) 2024-04-17 EP claimed
EP-3122757-B1 CHARGED LINKERS AND THEIR USES FOR CONJUGATION HANGZHOU DAC BIOTECH CO LTD (CN) 2023-09-06 EP claimed
EP-3845253-B1 SUSTAINED-RELEASE INJECTION PREPARATION CONTAINING CONJUGATE OF POLY-L-LACTIC ACID FILLER AND HYALURONIC ACID FILLER AND MANUFACTURING METHOD THEREFOR GCS CO LTD (KR) 2023-03-22 EP claimed
EP-3021832-B9 PRESERVED ETHERIFIED CYCLODEXTRIN DERIVATIVES CONTAINING LIQUID AQUEOUS PHARMACEUTICAL COMPOSITION BOEHRINGER INGELHEIM VETMEDICA GMBH (DE) 2023-03-15 EP claimed
EP-1227856-A1 INHALATION NEBULIZER PARI GmbH Spezialisten für effektive Inhalation (DE) 2002-08-07 EP claimed
WO-2001034232-A9 INHALATION NEBULIZER PARI GMBH (DE) 2002-08-01 WO claimed
EP-0925308-B1 COMPOSITIONS AND METHODS FOR TREATING INFECTIONS USING ANALOGUES OF INDOLICIDIN MICROLOGIX BIOTECH INC (CA) 2002-06-05 EP claimed
EP-1115405-A1 USE OF CERTAIN DRUGS FOR TREATING NERVE ROOT INJURY A+ Science Invest AB (SE) 2001-07-18 EP claimed
WO-2001034232-A1 INHALATION NEBULIZER Pari GmbH Spezialisten für effektive Inhalation (DE) 2001-05-17 WO claimed
EP-0661974-B1 METHODS AND COMPOSITIONS FOR TREATING INFECTION USING OPTICALLY PURE (R)-LOMEFLOXACIN SEPRACOR INC (US) 2000-09-06 EP claimed
WO-2000018409-A1 USE OF CERTAIN DRUGS FOR TREATING NERVE ROOT INJURY A+ SCIENCE INVEST AB (SE) 2000-04-06 WO claimed
EP-0659763-B1 21-Hydroxy pregnane - Quinoline carboxylic acid esters and Antibacterial and Antiinflammatory compositions containing them SENJU PHARMA CO (JP) 1998-05-20 EP claimed
EP-0443381-B2 Effervescent composition, its production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-10-22 EP claimed
EP-0394553-B1 Use of fluorine containing pyridone carboxylic acid derivatives for preparing a medicament for the treatment of HIV infections DAIICHI SEIYAKU CO (JP) 1995-06-21 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260027140-A1 COMPOSITIONS AND METHODS FOR TREATING AND AMELIORATING RESPIRATORY CONDITIONS AND INFLAMMATION OF MUCOSA IL1B, IL5, SERPINB1 KDM4E 4014/4885HSD17B10 3520/4885ALDH1A1 4294/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.