SCHEMBL13405754

SCHEMBL13405754

CC1CCN(c2nc(N3CCN(CC(=O)N4CCOCC4)CC3)ccc2NC(=O)c2ccc(C#N)o2)CC1

nearest known ligand 0.72

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 18/20 0.72
KDM4E B2RXH2 2/20 0.45
ALDH1A1 P00352 2/20 0.45
GAA P10253 1/20 0.45
RECQL P46063 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13405756 0.97 CSF1R (0.72) CSF1RKDM4EALDH1A1GAARECQL
Trifluoroacetic Acid SCHEMBL3540848 0.92 CSF1R (0.66) CSF1RKDM4EALDH1A1GAA
SCHEMBL3969432 0.88 CSF1R (0.56) CSF1RKDM4EALDH1A1GAARECQL
SCHEMBL13767720 0.86 CSF1R (0.56) CSF1RKDM4EALDH1A1GAARECQL
SCHEMBL13405733 0.84 CSF1R (1.00) CSF1R
SCHEMBL3544978 0.79 CSF1R (0.79) CSF1R
SCHEMBL13405752 0.79 CSF1R (0.68) CSF1R
SCHEMBL3534730 0.77 ALDH1A1 (0.50) CSF1RKDM4EALDH1A1RECQL
SCHEMBL5188971 0.75 ALDH1A1 (0.55) KDM4EALDH1A1GAARECQL
SCHEMBL3537014 0.74 MAPT (0.48) KDM4EALDH1A1GAARECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7705042-B2 Class of arylamide compounds useful as inhibitors of c-fms kinase JANSSEN PHARMACEUTICA NV (BE) 2010-04-27 US disclosed
US-7705042-B2 Class of arylamide compounds useful as inhibitors of c-fms kinase JANSSEN PHARMACEUTICA NV (BE) 2010-04-27 US disclosed