SCHEMBL1342

SCHEMBL1342

OCc1cn(C(c2ccccc2)(c2ccccc2)c2ccccc2)cn1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 15/20 0.45
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
ENPP2 Q13822 1/20 0.39
NOTUM Q6P988 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
NMBR P28336 1/20 0.36
P2RX7 Q99572 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6771514 0.98 SIRT2 (0.44) SIRT2CYP11B1CYP11B2ENPP2NOTUM
Acetic Acid SCHEMBL7659782 0.92 SIRT2 (0.47) SIRT2CYP11B1CYP11B2ENPP2NOTUM
SCHEMBL9069663 0.87 SIRT2 (0.44) SIRT2P2RX7
SCHEMBL1041048 0.87 SIRT2 (0.49) SIRT2CYP11B1CYP11B2ENPP2NMBR
SCHEMBL7713289 0.84 SIRT2 (0.46) SIRT2NMBR
SCHEMBL7939506 0.84 SIRT2 (0.40) SIRT2CYP11B1CYP11B2ENPP2NMBR
SCHEMBL2032778 0.84 SIRT2 (0.47) SIRT2CYP11B1CYP11B2ENPP2NMBR
SCHEMBL4682888 0.83 SIRT2 (0.46) SIRT2CYP11B1CYP11B2ENPP2NMBR
SCHEMBL1924923 0.83 SIRT2 (0.45) SIRT2CYP11B1CYP11B2ENPP2NOTUM
SCHEMBL2038903 0.83 SIRT2 (0.45) SIRT2CYP11B1CYP11B2ENPP2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 377 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760811-A1 IMIDAZOLE DERIVATIVES AS HISTAMINE RECEPTOR H 3? (ANT)AGONISTS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 1997-03-12 EP claimed
JP-1294682-A None JP disclosed
EP-4630424-A1 COMPOUNDS AND COMPOSITIONS AS C-KIT KINASE INHIBITORS Third Harmonic Bio, Inc. (US) 2025-10-15 EP disclosed
US-20250197368-A1 2-OXO-DIHYDROQUINOLINE-3-CARBOXAMIDE DERIVATIVES AS GABA TYPE A RECEPTOR MODULATORS DRAIG THERAPEUTICS LTD. (GB) 2025-06-19 US disclosed
US-12281101-B2 Bicyclic lactams and methods of use thereof GENENTECH, INC. (US) 2025-04-22 US disclosed
WO-2024240240-A1 IMIDAZOLE DERIVATIVES, INTERMEDIATE, PREPARATION METHOD THEREFOR AND USE THEREOF 江苏恩华药业股份有限公司 2024-11-28 WO disclosed
CN-118994283-A Beta-D-galactopyranose compound, preparation method, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2024-11-22 CN disclosed
CN-118684633-A Androgen receptor modulators and methods of use thereof 埃萨制药股份有限公司 2024-09-24 CN disclosed
US-20240254119-A1 COMPOUNDS AND COMPOSITIONS AS c-Kit KINASE INHIBITORS Calixis Inc. 2024-08-01 US disclosed
CN-113195441-B Androgen receptor modulators and methods of use thereof 埃萨制药股份有限公司 2024-07-12 CN disclosed
US-5026722-A Antagonists of 5-hydroxytryptamine GLAXO GROUP LIMITED (GB) 1991-06-25 US disclosed
EP-0383281-A1 1,2-ethanediol derivative and salt thereof, process for producing the same, and cerebral function-improving agent comprising the same TOYAMA CHEMICAL CO., LTD. (JP) 1990-08-22 EP disclosed
EP-0369743-A2 Heterocyclic amides ZENECA LIMITED (GB) 1990-05-23 EP disclosed
JP-H01294682-A PRODUCTION OF PHOSPHATIDYLCHOLINE NIPPON OIL & FATS CO LTD 1989-11-28 JP disclosed
US-4882343-A ADRENERGIC BLOCKING AGENTS G. D. SEARLE & CO. (US) 1989-11-21 US disclosed
EP-0338939-A1 Histamine derivative, process for his preparation and his therapeutic application INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 1989-10-25 EP disclosed
US-4814343-A ANTIISCHEMIC U C B, S.A. (BE) 1989-03-21 US disclosed
EP-0306323-A2 Lactam derivatives GLAXO GROUP LIMITED (GB) 1989-03-08 EP disclosed
EP-0304910-A1 Biarylalkylimidazole derivatives as antidepressants G.D. Searle & Co. (US) 1989-03-01 EP disclosed
EP-0269599-A2 Substituted 1H-imidazoles U C B, S.A. (BE) 1988-06-01 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12281101-B2 Bicyclic lactams and methods of use thereof LSS, LPXN, CYP1B1 SIRT2 1787/4885CYP11B1 143/4885CYP11B2 399/4885
US-20240254119-A1 COMPOUNDS AND COMPOSITIONS AS c-Kit KINASE INHIBITORS KIT, AURKC, PRKCE SIRT2 4277/4885CYP11B1 4060/4885CYP11B2 4434/4885
US-20250197368-A1 2-OXO-DIHYDROQUINOLINE-3-CARBOXAMIDE DERIVATIVES AS GABA TYPE A RECEPTOR MODULATORS GABRA2, GABRA3, GABRB2 SIRT2 1384/4885CYP11B1 595/4885CYP11B2 395/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.