SCHEMBL1343517

SCHEMBL1343517

N#Cc1ccc(Br)c2ccccc12

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 3/20 0.52
IMPDH1 P20839 2/20 0.52
AR P10275 7/20 0.47
DYRK1A Q13627 1/20 0.44
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CYP19A1 P11511 1/20 0.39
TSHR P16473 1/20 0.38
NCOA3 Q9Y6Q9 1/20 0.38
SLC22A12 Q96S37 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30478001 0.86 DYRK1A (0.53) IMPDH2IMPDH1ARDYRK1AKDM4E
SCHEMBL1343833 0.86 DYRK1A (0.53) IMPDH2IMPDH1ARDYRK1AKDM4E
SCHEMBL29489135 0.85 IMPDH2 (0.64) IMPDH2IMPDH1ARKDM4EALDH1A1
SCHEMBL151936 0.85 IMPDH2 (0.64) IMPDH2IMPDH1ARKDM4EALDH1A1
SCHEMBL11193357 0.83 IMPDH2 (0.61) IMPDH2IMPDH1ARKDM4EALDH1A1
SCHEMBL11200010 0.81 IMPDH2 (0.55) IMPDH2IMPDH1ARKDM4EALDH1A1
SCHEMBL11228244 0.80 IMPDH2 (0.59) IMPDH2IMPDH1ARKDM4EALDH1A1
SCHEMBL16917824 0.78 IMPDH2 (0.57) IMPDH2IMPDH1ARKDM4EALDH1A1
SCHEMBL7207783 0.77 RXFP1 (0.40) IMPDH2IMPDH1KDM4EALDH1A1GAA
SCHEMBL14873787 0.77 RXFP1 (0.36) IMPDH2IMPDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 177 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118955327-A Synthesis method of 4-bromo-1-naphthalene carbonitrile 安徽大学 2024-11-15 CN claimed
CN-116813834-B Flexible stretchable organic room-temperature phosphorescent material and preparation method thereof 南京邮电大学 2023-11-14 CN claimed
CN-116813834-A Flexible stretchable organic room-temperature phosphorescent material and preparation method thereof 南京邮电大学 2023-09-29 CN claimed
CN-114133387-B Fluorescent probe with viscosity sensing property and capable of targeting multiple organelles 郑州大学 2023-04-07 CN claimed
CN-114874197-A Viscosity fluorescent probe capable of targeting various organelles 郑州大学 2022-08-09 CN claimed
CN-114133387-A Fluorescent probe with viscosity sensing property and capable of targeting multiple organelles 郑州大学 2022-03-04 CN claimed
CN-112724153-A Three lyotropic colorimetric/lyotropic fluorescent probes with dual mitochondrial/lysosomal targeting 郑州大学 2021-04-30 CN claimed
CN-109734671-B Benzimidazole derivative, preparation method and application thereof 北京医药集团有限责任公司 2021-03-09 CN claimed
CN-107400090-B Synthesis method of benzimidazole derivative 华润赛科药业有限责任公司 2020-02-07 CN claimed
EP-4126835-B1 INHIBITORS OF ANTIGEN PRESENTATION BY HLA-DR JANSSEN PHARMACEUTICA NV (BE) 2026-02-18 EP disclosed
US-12516038-B2 Inhibitors of antigen presentation by HLA-DR JANSSEN PHARMACEUTICA NV (BE) 2026-01-06 US disclosed
US-20250346587-A1 NITROGEN-CONTAINING FIVE-MEMBERED HETEROCYCLIC DERIVATIVES AS CHECKPOINT KINASE 1 INHIBITOR AND USES THEREOF SPEROGENIX THERAPEUTICS LTD (CN) 2025-11-13 US disclosed
US-20250289826-A1 PLPRO PROTEIN INHIBITOR, AND PREPARATION METHOD AND APPLICATION THEREOF TSINGHUA UNIVERSITY (CN) 2025-09-18 US disclosed
WO-2025135309-A1 ORGANIC LIGHT-EMITTING COMPOUND, AND ORGANIC ELECTROLUMINESCENT DEVICE COMPRISING SAME 솔루스첨단소재 주식회사 2025-06-26 WO disclosed
US-20040180235-A1 Fluorescent diketopyrrolopyrroles CIBA SPECIALTY CHEMICALS CORP. 2004-09-16 US disclosed
US-20040122001-A1 Pharmaceutical compounds ELI LILLY AND COMPANY 2004-06-24 US disclosed
EP-1399514-A2 FLUORESCENT DIKETOPYRROLOPYRROLES Ciba SC Holding AG (CH) 2004-03-24 EP disclosed
EP-1345930-A2 PHARMACEUTICAL COMPOUNDS ELI LILLY AND COMPANY (US) 2003-09-24 EP disclosed
WO-2003002672-A2 FLUORESCENT DIKETOPYRROLOPYRROLES CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2003-01-09 WO disclosed
WO-2002050067-A2 PHARMACEUTICAL HETEROCYCLIC COMPOUNDS ELI LILLY AND COMPANY (US) 2002-06-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250346587-A1 NITROGEN-CONTAINING FIVE-MEMBERED HETEROCYCLIC DERIVATIVES AS CHECKPOINT KINASE 1 INHIBITOR AND USES THEREOF CHEK1, CHEK2, BUB1 IMPDH2 717/4885IMPDH1 458/4885AR 2944/4885
US-20040180235-A1 Fluorescent diketopyrrolopyrroles TYR, QDPR, PDK1 IMPDH2 942/4885IMPDH1 920/4885AR 3635/4885
US-20040122001-A1 Pharmaceutical compounds CYP2D6, LPXN, CYP1B1 IMPDH2 3369/4885IMPDH1 2164/4885AR 607/4885
US-20250289826-A1 PLPRO PROTEIN INHIBITOR, AND PREPARATION METHOD AND APPLICATION THEREOF ACE, PLP2, ACE2 IMPDH2 2418/4885IMPDH1 1940/4885AR 3631/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.