SCHEMBL13440433

SCHEMBL13440433

O=C1NS(=O)(=O)c2c(CBr)cccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 7/20 0.46
CA9 Q16790 7/20 0.46
CA2 P00918 5/20 0.46
CA7 P43166 4/20 0.46
CA1 P00915 3/20 0.46
KDM4E B2RXH2 1/20 0.46
USP2 O75604 1/20 0.46
LMNA P02545 1/20 0.46
BCHE P06276 1/20 0.46
CA4 P22748 1/20 0.46
CA6 P23280 1/20 0.46
CA5A P35218 1/20 0.46
KMT2A Q03164 1/20 0.46
CA14 Q9ULX7 1/20 0.46
CA5B Q9Y2D0 1/20 0.46
PDE7A Q13946 2/20 0.37
PDE7B Q9NP56 1/20 0.37
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL529430 0.80 CA12 (0.43) CA12CA9CA2CA7CA1
SCHEMBL82972 0.79 GABRA1 (0.45) CA12CA9CA2CA7CA1
SCHEMBL3807234 0.79 CA12 (0.46) CA12CA9CA2CA7CA1
SCHEMBL3806455 0.78 PTGER4 (0.47) CA12CA9CA2CA7CA1
SCHEMBL504060 0.76 NR1H2 (0.43) CA12CA9CA2CA7CA1
SCHEMBL3417559 0.75 NR1H2 (0.46) CA12CA9CA2CA7CA1
SCHEMBL9751229 0.75 NR1H2 (0.46) CA12CA9CA2CA7CA1
SCHEMBL14958500 0.74 CA12 (0.39) CA12CA9CA2CA7CA1
SCHEMBL9179277 0.73 RET (0.53) CA12CA9CA2CA7CA1
SCHEMBL995389 0.73 CA12 (0.50) CA12CA9CA2CA7CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7674810-B2 1,1-dioxo-1H-1Λ6-benzo[d]isothiazol-3-yl)-4-hydroxy-1,5-dihydro-pyrrol-2-one inhibitors of HCV polymerase ROCHE PALO ALTO LLC (US) 2010-03-09 US disclosed
US-7674810-B2 1,1-dioxo-1H-1Λ6-benzo[d]isothiazol-3-yl)-4-hydroxy-1,5-dihydro-pyrrol-2-one inhibitors of HCV polymerase ROCHE PALO ALTO LLC (US) 2010-03-09 US disclosed