SCHEMBL13452964

SCHEMBL13452964

C[C@@H]1CC=c2ccccc2=N1

nearest known ligand 0.32

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.32
NOS2 P35228 1/20 0.32
NISCH Q9Y2I1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13355549 1.00 NOS3 (0.32) NOS3NOS2NISCH
SCHEMBL10057749 1.00 NOS3 (0.32) NOS3NOS2NISCH
SCHEMBL13157598 0.75
SCHEMBL20219274 0.75
SCHEMBL19360573 0.72 CCR2 (0.33) NISCH
SCHEMBL28807372 0.72 TAAR1 (0.42) NOS3NOS2
SCHEMBL14147152 0.71 GSK3B (0.30)
SCHEMBL10111693 0.69
SCHEMBL28406757 0.68 HTR2B (0.41)
SCHEMBL6369641 0.65 NISCH (0.34) NOS3NOS2NISCH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1966191-B1 SUBSTITUTED PYRAZINONE DERIVATIVES AS ALPHA2C-ADRENORECEPTOR ANTAGONISTS JANSSEN PHARMACEUTICA NV (BE) 2010-03-17 EP disclosed