SCHEMBL134538

SCHEMBL134538

CN1OCC(=O)N(c2cccc(C(F)(F)F)c2)C1=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
AR P10275 1/20 0.49
CYP1A2 P05177 1/20 0.45
HTT P42858 1/20 0.45
ALDH1A1 P00352 4/20 0.44
TSHR P16473 1/20 0.44
DRD2 P14416 1/20 0.43
DRD3 P35462 1/20 0.43
ELANE P08246 4/20 0.42
CYP3A4 P08684 2/20 0.42
ALOX5 P09917 1/20 0.42
KDM4E B2RXH2 1/20 0.42
USP2 O75604 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
ALOX15 P16050 1/20 0.42
ALOX12 P18054 1/20 0.42
RECQL P46063 1/20 0.42
HSD17B10 Q99714 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29396063 1.00 MEN1 (0.52) MEN1KMT2AARCYP1A2HTT
SCHEMBL4887099 1.00 MEN1 (0.52) MEN1KMT2AARCYP1A2HTT
SCHEMBL11278353 0.78 MEN1 (0.56) MEN1KMT2AARCYP1A2ALDH1A1
SCHEMBL28744553 0.77 MEN1 (0.70) MEN1KMT2AARCYP1A2HTT
SCHEMBL29702930 0.77 MEN1 (0.70) MEN1KMT2AARCYP1A2HTT
SCHEMBL15837517 0.77 MEN1 (0.62) MEN1KMT2AARCYP1A2HTT
SCHEMBL10344670 0.73 MEN1 (0.45) MEN1KMT2AHTTALDH1A1TSHR
SCHEMBL11281751 0.72 DRD2 (0.52) MEN1KMT2AARCYP1A2ALDH1A1
SCHEMBL17047686 0.71 AR (0.57) MEN1KMT2AARCYP1A2HTT
SCHEMBL3180022 0.71 MGLL (0.64) MEN1KMT2AARCYP1A2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3747 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3060043-B1 PESTICIDAL COMPOSITIONS AND RELATED METHODS CORTEVA AGRISCIENCE LLC (US) 2025-11-26 EP claimed
EP-3578542-B1 COMPOSITIONS HAVING PESTICIDAL UTILITY AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-11-12 EP claimed
EP-3578543-B1 COMPOSITIONS COMPRISING MOLECULES HAVING PESTICIDAL UTILITY AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-08-20 EP claimed
US-20250176551-A1 METHOD FOR CONTROLLING THE GROWTH OF UNDESIRABLE VEGETATION UPL LTD (IN) 2025-06-05 US claimed
EP-3578541-B1 COMPOSITIONS COMPRISING MOLECULES HAVING PESTICIDAL UTILITY, AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-05-28 EP claimed
US-20250113826-A1 AN AGROCHEMICAL COMBINATION UPL LTD (IN) 2025-04-10 US claimed
US-20240172758-A1 METHOD FOR CONTROLLING THE GROWTH OF UNDESIRABLE VEGETATION UPL LIMITED (IN) 2024-05-30 US claimed
US-20230139897-A1 SOLID HERBICIDE COMPOSITION AND THE USE THEREOF ROTAM AGROCHEM INTERNATIONAL COMPANY LIMITED (HK) 2023-05-04 US claimed
WO-2023067621-A1 AN AGROCHEMICAL COMBINATION UPL LIMITED (IN) 2023-04-27 WO claimed
WO-2023062434-A1 A METHOD FOR CONTROLLING THE GROWTH OF UNDESIRABLE VEGETATION UPL LIMITED (IN) 2023-04-20 WO claimed
CN-1555219-A Herbicidal mixtures based on 3-phenyluracils �����ɷ� 2004-12-15 CN claimed
US-20040235665-A1 used in combination with other herbicides and possibly plant safening agents in order to reduce toxic effect on plants BASF AKTIENGESELLSCHAFT (DE) 2004-11-25 US claimed
EP-1458237-A1 HERBICIDAL MIXTURE BASED ON 7-PYRAZOLYLBENZOXAZOLES BASF AKTIENGESELLSCHAFT (DE) 2004-09-22 EP claimed
EP-1429609-A1 HERBICIDAL MIXTURES BASED ON 3-PHENYLURACILS BASF AKTIENGESELLSCHAFT (DE) 2004-06-23 EP claimed
US-6683027-B2 SYNERGISTICALLY EFFECTIVE AMOUNT OF SUBSTITUTED 2-PHENYL PYRIMIDINE COMPOUNDS WITH OTHER HERBICIDAL COMPOUND, WHICH IS ACTIVE AGAINST BROAD-LEAVED WEEDS AND/OR ANNUAL GRASSES BASF AKTIENEGESELLSCHAFT (DE) 2004-01-27 US claimed
WO-2003051122-A1 HERBICIDAL MIXTURE BASED ON 7-PYRAZOLYLBENZOXAZOLES BASF AKTIENGESELLSCHAFT (DE) 2003-06-26 WO claimed
EP-1313369-A2 HERBICIDAL MIXTURES BASF AKTIENGESELLSCHAFT (DE) 2003-05-28 EP claimed
WO-2003024221-A1 HERBICIDAL MIXTURES BASED ON 3-PHENYLURACILS BASF AKTIENGESELLSCHAFT (DE) 2003-03-27 WO claimed
US-20020055435-A1 Herbicidal mixtures INTELLECTUAL PROPERTY DEPARTMENT (DE) 2002-05-09 US claimed
WO-2002015694-A2 HERBICIDAL MIXTURES BASF AKTIENGESELLSCHAFT (DE) 2002-02-28 WO claimed