SCHEMBL13458285

SCHEMBL13458285

C1=NC(c2cnc(-c3ccccc3)nc2)CN1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.44
RAB9A P51151 4/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
NFKB1 P19838 2/20 0.44
NFKB2 Q00653 2/20 0.44
RELA Q04206 2/20 0.44
HTR2C P28335 1/20 0.40
HPGDS O60760 11/20 0.40
MAPK1 P28482 1/20 0.36
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
RECQL P46063 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11545883 0.79 SLC18A3 (0.39) HTR2CLMNA
SCHEMBL13457870 0.69 NPC1 (0.46) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL13458139 0.68 NPC1 (0.44) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL13458303 0.67 NPC1 (0.43) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL11547375 0.65 SLC6A3 (0.44) LMNA
SCHEMBL40296 0.64 RAB9A (0.65) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL2117282 0.64 NPC1 (1.00) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL13457849 0.64 NISCH (0.50) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL14044884 0.63 DRD3 (0.46) HTR2CLMNA
SCHEMBL12647379 0.63 KDM1A (0.47) HTR2CLMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010033977-A2 MULTIHETEROARYL COMPOUNDS AS INHIBITORS OF H-PGDS AND THEIR USE FOR TREATING PROSTAGLANDIN D2 MEDIATED DISEASES CAYMAN CHEMICAL COMPANY (US) 2010-03-25 WO disclosed