SCHEMBL11545883

SCHEMBL11545883

C1=NC(c2ccccc2)CN1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC18A3 Q16572 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
TAAR1 Q96RJ0 3/20 0.37
MAOB P27338 8/20 0.37
MAOA P21397 7/20 0.37
KDM1A O60341 5/20 0.37
CYP2C19 P33261 4/20 0.37
CYP2B6 P20813 3/20 0.37
CYP1A2 P05177 2/20 0.37
CYP2D6 P10635 2/20 0.37
CYP2C9 P11712 2/20 0.37
LMNA P02545 2/20 0.37
CYP3A4 P08684 1/20 0.37
HTR1A P08908 1/20 0.37
ADRA2A P08913 1/20 0.37
CYP2A6 P11509 1/20 0.37
SLC6A2 P23975 1/20 0.37
HTR2C P28335 1/20 0.37
ADRA1A P35348 1/20 0.37
DRD3 P35462 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17734079 0.81 CYP1A2 (0.34) CYP2C19CYP1A2LMNAHSD17B10
SCHEMBL11547375 0.79 SLC6A3 (0.44) TAAR1MAOBKDM1ALMNASLC6A2
SCHEMBL11094591 0.79 SLC18A3 (0.41) SLC18A3SIGMAR1TAAR1MAOBMAOA
SCHEMBL13458285 0.79 NPC1 (0.44) LMNAHTR2C
SCHEMBL14044884 0.77 DRD3 (0.46) KDM1ALMNACYP3A4HTR2CDRD3
SCHEMBL12647379 0.77 KDM1A (0.47) KDM1ALMNAHTR2CRCOR1
SCHEMBL11828815 0.75
SCHEMBL4559809 0.75 CYP11B2 (0.38) KDM1ACYP2A6KCNH2
SCHEMBL11835500 0.75 ALDH1A1 (0.35) CYP2A6CYP2A13HSD17B10
SCHEMBL11286867 0.74 MAOB (0.38) TAAR1MAOBMAOAKDM1ACYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109311903-A Cyclic annular 3- phenyl tetramic acid derivatives with herbicide effect 拜耳作物科学股份公司 2019-02-05 CN disclosed
EP-3194406-A1 TRICYCLIC HETEROCYCLES FOR USE AS BET PROTEIN INHIBITORS Incyte Holdings Corporation (US) 2017-07-26 EP disclosed
WO-2016044130-A1 TRICYCLIC HETEROCYCLES FOR USE AS BET PROTEIN INHIBITORS INCYTE CORPORATION (US) 2016-03-24 WO disclosed
CN-1004272-B PYRAZOLINE INSECTICIDES FMC公司 1989-05-24 CN disclosed
US-4163857-A DRUGS, FUNGICIDES BAYER AKTIENGESELLSCHAFT (DE) 1979-08-07 US disclosed
US-4105765-A ANTITHROMBOTICS, ANTICOAGULANTS BOEHRINGER INGELHEIM GMBH (DE) 1978-08-08 US disclosed
US-4058616-A ANTITHROMBOTICS BOEHRINGER INGELHEIM GMBH (DT) 1977-11-15 US disclosed
US-3966801-A ANTIINFLAMMATORY AGENTS WILLIAM H. RORER, INC. (US) 1976-06-29 US disclosed