SCHEMBL13465305

SCHEMBL13465305

N#Cc1ccc(CCC2(c3ccncc3)CCC(=O)NC2=O)cc1

nearest known ligand 0.60

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 19/20 0.60
ALDH1A1 P00352 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17898240 0.81 CYP19A1 (0.38) CYP19A1CYP2D6
SCHEMBL3296751 0.74 CYP19A1 (1.00) CYP19A1
Rogletimide SCHEMBL9372682 0.73 CYP19A1 (1.00) CYP19A1
Rogletimide SCHEMBL4281 0.73 CYP19A1 (1.00) CYP19A1
SCHEMBL9531145 0.72 CYP19A1 (1.00) CYP19A1
Rogletimide SCHEMBL28110686 0.71 CYP19A1 (0.94) CYP19A1
SCHEMBL10514138 0.70 CYP19A1 (0.68) CYP19A1
SCHEMBL20805215 0.65 CYP19A1 (0.60) CYP19A1
SCHEMBL171234 0.60 HRH3 (0.53) CYP19A1ALDH1A1CYP1A2CYP2D6
SCHEMBL11847657 0.60 ALDH1A1 (0.54) CYP19A1ALDH1A1CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120265514-A1 DESIGN OF MOLECULES UNIVERSITY OF DUNDEE (GB) 2012-10-18 US disclosed