SCHEMBL17898240

SCHEMBL17898240

N#Cc1ccc(CCC2(c3ccncc3)CCS(=O)(=O)NC2=O)cc1

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 16/20 0.38
SMN1; SMN2 Q16637 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2D6 P10635 1/20 0.35
MMP13 P45452 2/20 0.34
GAA P10253 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13465305 0.81 CYP19A1 (0.60) CYP19A1CYP2D6
SCHEMBL171234 0.58 HRH3 (0.53) CYP19A1CYP3A4CYP2D6
SCHEMBL1004267 0.57 LOXL2 (0.64) CYP19A1MMP13
SCHEMBL9127449 0.56 MAOB (0.60) CYP19A1SMN1; SMN2CYP3A4GAARAB9A
Isonicotinonitrile SCHEMBL12264099 0.55
Isonicotinonitrile SCHEMBL2015834 0.55 HDAC8 (0.52) CYP19A1GAA
Isonicotinonitrile SCHEMBL151611 0.55
Isonicotinonitrile SCHEMBL28123141 0.55 ADRB2 (0.43)
SCHEMBL8390135 0.55 LOXL2 (0.54) CYP19A1MMP13
SCHEMBL508063 0.55 LOXL2 (0.54) CYP19A1MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10381110-B2 Molecules UNIVERSITY OF DUNDEE (GB) 2019-08-13 US disclosed
US-20160196412-A1 DESIGN OF MOLECULES RECURSION PHARMACEUTICALS, INC. 2016-07-07 US disclosed
US-20160196412-A1 DESIGN OF MOLECULES RECURSION PHARMACEUTICALS, INC. 2016-07-07 US disclosed