SCHEMBL13475017

SCHEMBL13475017

CCCCc1ccc(N(c2ccccc2)c2ccc(N(c3ccc(C(C)CC)cc3)c3ccc(N(c4ccccc4)c4ccc(CCCC)cc4)cc3)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.47
KCNH2 Q12809 2/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
HSD11B1 P28845 1/20 0.40
CHRM2 P08172 1/20 0.40
HTR1A P08908 1/20 0.40
ADRA2A P08913 1/20 0.40
CHRM1 P11229 1/20 0.40
DRD1 P21728 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
ADRA1A P35348 1/20 0.40
OPRM1 P35372 1/20 0.40
DRD3 P35462 1/20 0.40
SLC6A3 Q01959 1/20 0.40
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
BCHE P06276 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18494830 0.96 HSD11B1 (0.43) HTR2ACA1CA2HSD11B1ALDH1A1
SCHEMBL17986526 0.94 HTR2A (0.55) HTR2AKCNH2HSD11B1CHRM2ADRA2A
SCHEMBL25907712 0.89 UCHL3 (0.45) HTR2ACA1CA2ALDH1A1HPGD
SCHEMBL12018269 0.89 UCHL3 (0.45) HTR2ACA1CA2ALDH1A1HPGD
SCHEMBL15854779 0.88 CA1 (0.40) HTR2AKCNH2CA1CA2ALDH1A1
SCHEMBL13474932 0.87 NPC1 (0.41) HTR2ACA1CA2ALDH1A1HPGD
SCHEMBL14292089 0.87 GPR88 (0.41) HTR2ASIGMAR1
SCHEMBL13474954 0.85 SMN1; SMN2 (0.43) CA1CA2ALDH1A1HPGD
SCHEMBL10042891 0.85 KCNH2 (0.52) HTR2AKCNH2CA1CA2HSD11B1
SCHEMBL987390 0.85 KCNH2 (0.52) HTR2AKCNH2CA1CA2HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7666956-B2 Polymer MERCK PATENT GMBH (DE) 2010-02-23 US disclosed
US-7666956-B2 Polymer MERCK PATENT GMBH (DE) 2010-02-23 US disclosed