SCHEMBL13486346

SCHEMBL13486346

CCc1ccc(Oc2ccc(C(C)=O)cc2F)c(OC(=O)CNCl)c1

nearest known ligand 0.63

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 1/20 0.39
TMPRSS15 P98073 1/20 0.39
AKT1 P31749 1/20 0.37
TAS1R3 Q7RTX0 1/20 0.36
TAS1R1 Q7RTX1 1/20 0.36
CARM1 Q86X55 1/20 0.36
PRMT6 Q96LA8 1/20 0.36
ALOX15 P16050 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13486214 0.85 PRSS1 (0.41) PRSS1TMPRSS15CARM1PRMT6ALOX15
SCHEMBL3204847 0.85 EPHX2 (0.38) PRSS1TMPRSS15CARM1PRMT6
SCHEMBL3209730 0.81 LMNA (0.49) TAS1R3TAS1R1
SCHEMBL3201265 0.78
SCHEMBL3204839 0.76 PRSS1 (0.36) PRSS1TMPRSS15CARM1PRMT6ALOX15
SCHEMBL3212402 0.76 BRD4 (0.48)
Hydrochloric Acid SCHEMBL3191227 0.76 PTGDR (0.39) PRSS1TMPRSS15
Hydrochloric Acid SCHEMBL3191222 0.73 PTGDR (0.37) PRSS1TMPRSS15CARM1PRMT6
SCHEMBL27936118 0.71 SMN1; SMN2 (0.54)
SCHEMBL3214638 0.71 MAPK1 (0.53)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8722746-B2 Hydroxyphenyl derivatives and biological applications thereof FAB PHARMA S.A.S. (FR) 2014-05-13 US disclosed
US-20100041658-A1 Hydroxyphenyl Derivatives and Biological Applications Thereof FAB PHARMA (FR) 2010-02-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100041658-A1 Hydroxyphenyl Derivatives and Biological Applications Thereof HPD, HPGDS, EPX PRSS1 2000/4885TMPRSS15 545/4885AKT1 4283/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.