SCHEMBL13487155

SCHEMBL13487155

CCc1ccc2cc(N(C)C)ccc2c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.57
CYP2A6 P11509 1/20 0.57
APP P05067 3/20 0.47
TERT O14746 1/20 0.47
ALDH1A1 P00352 2/20 0.46
TSHR P16473 2/20 0.46
CYP3A4 P08684 1/20 0.46
MAPK1 P28482 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
PSMB5 P28074 2/20 0.46
AKR1C3 P42330 1/20 0.42
AKR1C2 P52895 1/20 0.42
CALM1 P0DP23 2/20 0.42
SIGMAR1 Q99720 1/20 0.42
ALOX15 P16050 1/20 0.40
HSD17B10 Q99714 1/20 0.40
TRPA1 O75762 1/20 0.39
EGFR P00533 2/20 0.38
NOS1 P29475 3/20 0.37
NOS2 P35228 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25085593 0.94 CYP1A2 (0.55) CYP1A2CYP2A6APPTERTALDH1A1
SCHEMBL15131776 0.84 SIGMAR1 (0.47) CYP1A2CYP2A6APPTERTALDH1A1
SCHEMBL347592 0.82 CYP2A6 (0.80) CYP1A2CYP2A6ALDH1A1MAPK1AKR1C3
SCHEMBL12566471 0.82 TERT (0.64) APPTERTALDH1A1TSHRCYP3A4
SCHEMBL29407167 0.82 CYP2A6 (0.80) CYP1A2CYP2A6ALDH1A1MAPK1AKR1C3
SCHEMBL14311184 0.82 APP (0.45) CYP2A6APPTERTALDH1A1TSHR
SCHEMBL6044185 0.82 APP (0.49) CYP1A2CYP2A6APPTERTALDH1A1
SCHEMBL1901448 0.80 SIGMAR1 (0.51) ALDH1A1CYP3A4SIGMAR1HSD17B10EGFR
SCHEMBL14311185 0.79 SIGMAR1 (0.46) CYP1A2CYP2A6APPTERTALDH1A1
SCHEMBL13432618 0.79 CYP1A2 (0.74) CYP1A2CYP2A6AKR1C3AKR1C2SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021118727-A2 FLUOROGENIC AMINO ACIDS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2021-06-17 WO disclosed
US-20130190497-A1 FLUORESCENT SUBSTRATES FOR MONOAMINE TRANSPORTERS AS OPTICAL FALSE NEUROTRANSMITTERS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2013-07-25 US disclosed
US-20100048604-A1 Ligands for Aldoketoreductases TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2010-02-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100048604-A1 Ligands for Aldoketoreductases AKR1C2, AKR1C1, AKR1B1 CYP1A2 98/4885CYP2A6 315/4885APP 3894/4885
US-20130190497-A1 FLUORESCENT SUBSTRATES FOR MONOAMINE TRANSPORTERS AS OPTICAL FALSE NEUROTRANSMITTERS SLC18A2, SLC6A2, SLC18A3 CYP1A2 1053/4885CYP2A6 1899/4885APP 1119/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.