SCHEMBL13541908

SCHEMBL13541908

CBc1cnn(CCN2CCCC2)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 3/20 0.37
JAK3 P52333 3/20 0.37
JAK1 P23458 1/20 0.37
TYK2 P29597 1/20 0.37
HRH3 Q9Y5N1 4/20 0.36
SIGMAR1 Q99720 5/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
FGFR1 P11362 1/20 0.35
FGFR2 P21802 1/20 0.35
FGFR4 P22455 1/20 0.35
FGFR3 P22607 1/20 0.35
KDR P35968 1/20 0.35
FLT3 P36888 1/20 0.35
PTK2 Q05397 2/20 0.34
TERT O14746 1/20 0.33
KMT2A Q03164 1/20 0.33
MET P08581 1/20 0.33
HRH4 Q9H3N8 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11946810 0.79 HRH3 (0.42) JAK2JAK3JAK1TYK2HRH3
SCHEMBL986124 0.79 CHRNB2 (0.36) JAK2JAK3JAK1TYK2HRH3
SCHEMBL17793165 0.77 HRH3 (0.41) JAK2JAK3JAK1TYK2HRH3
SCHEMBL2581848 0.77 TERT (0.38) JAK2JAK3JAK1TYK2HRH3
SCHEMBL17789616 0.76 MEN1 (0.43) JAK2JAK3JAK1TYK2SIGMAR1
SCHEMBL10263495 0.76 HRH3 (0.46) JAK2JAK3JAK1TYK2HRH3
SCHEMBL1703040 0.75 SIGMAR1 (0.41) JAK2JAK3JAK1TYK2HRH3
SCHEMBL10203212 0.75 KDM4E (0.43) JAK2JAK3JAK1TYK2HRH3
SCHEMBL10141504 0.75 MEN1 (0.42) JAK2JAK3JAK1TYK2SIGMAR1
SCHEMBL19267190 0.74 PSMB1 (0.34) JAK2JAK3JAK1TYK2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010000364-A1 PYRROLOPYRIDINYLPYRIMIDIN-2-YLAMINE DERIVATIVES MERCK PATENT GMBH (DE) 2010-01-07 WO disclosed