SCHEMBL13544009

SCHEMBL13544009

COc1cccc(N2CNC(=O)C23CCN(CCOC2(c4ccc(Cl)c(Cl)c4)CCN(C(=O)c4ccco4)CC2)CC3)c1

nearest known ligand 0.85

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 15/20 0.85
OPRK1 P41145 2/20 0.41
SLC6A3 Q01959 2/20 0.41
HTR1A P08908 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
HTR2C P28335 1/20 0.41
CACNA1F O60840 1/20 0.40
CHRM2 P08172 1/20 0.40
ADRB1 P08588 1/20 0.40
DRD2 P14416 1/20 0.40
SLC6A2 P23975 1/20 0.40
ADRA1D P25100 1/20 0.40
ADRA1A P35348 1/20 0.40
HRH1 P35367 1/20 0.40
ADRA1B P35368 1/20 0.40
OPRM1 P35372 1/20 0.40
DRD3 P35462 1/20 0.40
OPRD1 P41143 1/20 0.40
OPRL1 P41146 1/20 0.40
CACNA1D Q01668 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5511844 0.96 CCR5 (0.85) CCR5OPRK1SLC6A3HTR1AADORA3
SCHEMBL13544007 0.92 CCR5 (1.00) CCR5OPRK1ADORA3HTR2COPRM1
SCHEMBL13544013 0.89 CCR5 (0.66) CCR5OPRM1OPRL1
SCHEMBL4679383 0.88 CCR5 (1.00) CCR5OPRK1ADORA3HTR2COPRM1
SCHEMBL4679294 0.86 CCR5 (0.68) CCR5OPRM1OPRL1
SCHEMBL13544010 0.85 CCR5 (0.78) CCR5OPRK1HTR1AOPRM1OPRD1
SCHEMBL4685629 0.83 CCR5 (0.64) CCR5OPRM1OPRL1
SCHEMBL4682434 0.83 CCR5 (0.85) CCR5HTR1AOPRM1OPRL1
SCHEMBL6170250 0.82 CCR5 (0.63) CCR5OPRK1SLC6A3HTR1AADORA3
SCHEMBL13544014 0.81 CCR5 (0.86) CCR5OPRK1SLC6A3HTR1ACACNA1F

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7645771-B2 CCR5 antagonists as therapeutic agents SMITHKLINE BEECHAM CORP. (US) 2010-01-12 US disclosed