SCHEMBL13544014

SCHEMBL13544014

COc1cccc(N2CNC(=O)C23CCN(CCOC2(c4ccc(Cl)c(Cl)c4)CCN(S(=O)(=O)c4ccccc4)CC2)CC3)c1

nearest known ligand 0.86

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 13/20 0.86
OPRM1 P35372 3/20 0.46
OPRL1 P41146 3/20 0.46
HTR1A P08908 1/20 0.44
OPRD1 P41143 2/20 0.44
OPRK1 P41145 2/20 0.44
CACNA1F O60840 1/20 0.43
CHRM2 P08172 1/20 0.43
ADRB1 P08588 1/20 0.43
DRD2 P14416 1/20 0.43
SLC6A2 P23975 1/20 0.43
ADRA1D P25100 1/20 0.43
ADRA1A P35348 1/20 0.43
HRH1 P35367 1/20 0.43
ADRA1B P35368 1/20 0.43
DRD3 P35462 1/20 0.43
CACNA1D Q01668 1/20 0.43
SLC6A3 Q01959 1/20 0.43
CACNA1S Q13698 1/20 0.43
CACNA1C Q13936 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4686334 0.96 CCR5 (0.86) CCR5OPRM1OPRL1HTR1AOPRD1
SCHEMBL13544011 0.93 CCR5 (1.00) CCR5OPRM1OPRL1OPRD1OPRK1
SCHEMBL4683214 0.89 CCR5 (1.00) CCR5OPRM1OPRL1OPRD1OPRK1
SCHEMBL13544013 0.86 CCR5 (0.66) CCR5OPRM1OPRL1
SCHEMBL4679294 0.83 CCR5 (0.68) CCR5OPRM1OPRL1
SCHEMBL13544010 0.82 CCR5 (0.78) CCR5OPRM1OPRL1HTR1AOPRD1
SCHEMBL13544009 0.81 CCR5 (0.85) CCR5OPRM1OPRL1HTR1AOPRD1
SCHEMBL4685629 0.81 CCR5 (0.64) CCR5OPRM1OPRL1
SCHEMBL4682434 0.80 CCR5 (0.85) CCR5OPRM1OPRL1HTR1A
SCHEMBL6170250 0.80 CCR5 (0.63) CCR5OPRM1OPRL1HTR1AOPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7645771-B2 CCR5 antagonists as therapeutic agents SMITHKLINE BEECHAM CORP. (US) 2010-01-12 US disclosed