SCHEMBL13548601

SCHEMBL13548601

Cn1cc(Sc2ccccc2F)c2ccccc21

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 2/20 0.47
GPR84 Q9NQS5 1/20 0.43
HTR2A P28223 1/20 0.42
IMPDH2 P12268 2/20 0.41
RHEB Q15382 1/20 0.40
HTT P42858 1/20 0.40
BACE1 P56817 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MAPT P10636 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
NR4A2 P43354 1/20 0.37
IDO1 P14902 1/20 0.37
CCNE2 O96020 1/20 0.37
CDK4 P11802 1/20 0.37
CCND1 P24385 1/20 0.37
CCNE1 P24864 1/20 0.37
CDK2 P24941 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10221867 0.77 KDM4E (0.55) KDM4EALDH1A1GPR84HTR2AIMPDH2
SCHEMBL835657 0.76 KDM4E (0.53) KDM4EALDH1A1NPSR1MAPT
SCHEMBL21035552 0.76 GPR84 (0.57) KDM4EALDH1A1GPR84HTR2AIMPDH2
SCHEMBL1399520 0.75 ALDH1A1 (0.46) KDM4EALDH1A1GPR84HTR2AIMPDH2
SCHEMBL21027633 0.74 KDM4E (0.56) KDM4EALDH1A1GPR84HTR2AIMPDH2
SCHEMBL1399447 0.74 HTR2A (0.55) KDM4EALDH1A1GPR84HTR2AL3MBTL1
SCHEMBL1399471 0.74 LMNA (0.57) KDM4EALDH1A1
SCHEMBL17936381 0.73 MAPT (0.48) KDM4EALDH1A1GPR84IMPDH2HTT
SCHEMBL575956 0.73 HAO1 (0.52)
SCHEMBL28543725 0.72 KDM4E (0.50) KDM4EALDH1A1GPR84HTR2AIMPDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7645774-B2 Cannabinoid receptor ligands SCHERING CORPORATION (US) 2010-01-12 US disclosed
US-7645774-B2 Cannabinoid receptor ligands SCHERING CORPORATION (US) 2010-01-12 US disclosed