SCHEMBL13565261

SCHEMBL13565261

CCc1cc(NCCCCCNS(=O)(=O)C(C)(C)C)ccc1OC1CCCC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 3/20 0.40
NPY1R P25929 1/20 0.39
NPY2R P49146 1/20 0.39
RORC P51449 1/20 0.38
P2RX4 Q99571 1/20 0.36
POLB P06746 1/20 0.34
PDE4A P27815 3/20 0.34
FABP4 P15090 2/20 0.34
FABP5 Q01469 2/20 0.34
PDE4B Q07343 2/20 0.34
PDE4C Q08493 2/20 0.34
PDE4D Q08499 2/20 0.34
CYP19A1 P11511 2/20 0.33
EPHX2 P34913 2/20 0.33
LTB4R Q15722 1/20 0.33
PDE7A Q13946 1/20 0.33
MEN1 O00255 1/20 0.33
PTGES O14684 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13565176 0.85 HRH1 (0.41) CNR2NPY1RNPY2RRORCPOLB
SCHEMBL10115258 0.85 ALDH1A1 (0.46) RORCP2RX4POLBPDE4AMEN1
SCHEMBL11935716 0.82 CARM1 (0.38) NPY1RNPY2RRORCP2RX4POLB
SCHEMBL11935682 0.82 ACACB (0.38) CNR2RORCMEN1ALDH1A1MAPT
SCHEMBL13565527 0.81 CTSL (0.38) CNR2RORCEPHX2MEN1ALDH1A1
SCHEMBL13565836 0.81 HDAC4 (0.41) CNR2EPHX2
SCHEMBL13565477 0.80 HDAC4 (0.41) CNR2EPHX2ALDH1A1MAPT
SCHEMBL13566088 0.79 NPY1R (0.41) NPY1RNPY2RRORCP2RX4POLB
SCHEMBL13564791 0.75 CNR2 (0.39) CNR2POLBCYP19A1ALDH1A1MAPT
SCHEMBL13565263 0.75 CNR2 (0.48) CNR2POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed
US-8299265-B2 Amine derivatives having NPY Y5 receptor antagonistic activity and the uses thereof SHIONOGI & CO., LTD. (JP) 2012-10-30 US disclosed