SCHEMBL13565335

SCHEMBL13565335

Cc1ccc(NCc2ccc(NS(=O)(=O)C(C)C)cc2)c2c1CCCC2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.42
PPARA Q07869 1/20 0.36
GRIA2 P42262 1/20 0.36
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
RXRA P19793 1/20 0.35
RXRB P28702 1/20 0.35
RXRG P48443 1/20 0.35
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
CA9 Q16790 2/20 0.35
CA12 O43570 1/20 0.35
HDAC6 Q9UBN7 2/20 0.34
BRD4 O60885 1/20 0.34
ADRB2 P07550 2/20 0.34
ADRB1 P08588 2/20 0.34
ADRB3 P13945 1/20 0.34
METAP2 P50579 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11936096 0.84 PARP1 (0.42) PARP1PPARAGRIA2RXRARXRB
SCHEMBL13565080 0.83 RXRA (0.40) PARP1PPARAGRIA2HTTSMN1; SMN2
SCHEMBL13565505 0.83 SMN1; SMN2 (0.56) PARP1HTTSMN1; SMN2NPSR1RXRA
SCHEMBL13565355 0.82 METAP2 (0.35) HTTSMN1; SMN2NPSR1RXRARXRB
SCHEMBL10116637 0.78 LMNA (0.41) GRIA2HTTLMNATP53MAPT
SCHEMBL11936098 0.76 PARP1 (0.36) PARP1PPARACA1CA2CA9
SCHEMBL13565070 0.76 PPARA (0.50) PPARASMN1; SMN2CA1CA2BRD4
SCHEMBL13565984 0.76 CA1 (0.59) HTTSMN1; SMN2CA1CA2CA9
SCHEMBL11936110 0.75 PARP1 (0.37) PARP1GRIA2HTTSMN1; SMN2NPSR1
SCHEMBL17090103 0.75 ALDH1A1 (0.43) PPARASMN1; SMN2HDAC6LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed
US-8299265-B2 Amine derivatives having NPY Y5 receptor antagonistic activity and the uses thereof SHIONOGI & CO., LTD. (JP) 2012-10-30 US disclosed