SCHEMBL13565751

SCHEMBL13565751

CCC(C)S(=O)(=O)NC1CCC(CNc2ccc3ncccc3c2)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 1/20 0.44
ALDH1A1 P00352 2/20 0.40
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PIK3CD O00329 2/20 0.39
PIK3CA P42336 2/20 0.39
PIK3CB P42338 2/20 0.39
PIK3CG P48736 2/20 0.39
NPC1 O15118 2/20 0.39
MET P08581 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
POLB P06746 1/20 0.38
MAPT P10636 1/20 0.38
HDAC6 Q9UBN7 1/20 0.37
SYK P43405 2/20 0.37
MAT2A P31153 2/20 0.37
BRAF P15056 1/20 0.36
EPHX2 P34913 1/20 0.36
ULK1 O75385 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11936208 0.91 NR3C1 (0.46) NR3C1ALDH1A1LMNASMN1; SMN2PIK3CD
SCHEMBL13565664 0.91 NR3C1 (0.46) NR3C1ALDH1A1LMNASMN1; SMN2PIK3CD
SCHEMBL13565722 0.87 MET (0.43) ALDH1A1LMNASMN1; SMN2NPC1MET
SCHEMBL11936207 0.87 ALDH1A1 (0.43) NR3C1ALDH1A1LMNASMN1; SMN2PIK3CD
SCHEMBL11936220 0.83 NR3C1 (0.42) NR3C1ALDH1A1LMNASMN1; SMN2PIK3CD
SCHEMBL13565703 0.83 NR3C1 (0.42) NR3C1ALDH1A1LMNASMN1; SMN2PIK3CD
SCHEMBL10114221 0.83 EPHX2 (0.53) ALDH1A1LMNANPC1MEN1KMT2A
SCHEMBL17090186 0.80 IRAK4 (0.43) ALDH1A1IRAK4
SCHEMBL13565995 0.80 IRAK4 (0.43) ALDH1A1IRAK4
SCHEMBL13565025 0.78 BRD4 (0.39) ALDH1A1LMNASMN1; SMN2METMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed
US-8299265-B2 Amine derivatives having NPY Y5 receptor antagonistic activity and the uses thereof SHIONOGI & CO., LTD. (JP) 2012-10-30 US disclosed