SCHEMBL13565754

SCHEMBL13565754

CCC(C)S(=O)(=O)NC1CCC(CNc2ccc(Oc3ccccc3)cc2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.39
BACE1 P56817 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
NPY5R Q15761 2/20 0.39
PGR P06401 2/20 0.39
MAPT P10636 2/20 0.38
ALOX12 P18054 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HTT P42858 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
RECQL P46063 2/20 0.38
LMNA P02545 2/20 0.38
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
GFER P55789 1/20 0.37
EPHX2 P34913 1/20 0.36
HPGD P15428 1/20 0.36
MMP2 P08253 5/20 0.36
MMP13 P45452 5/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11935090 0.90 ACHE (0.41) ACHEBACE1NPY5RPGRMAPT
SCHEMBL13565599 0.85 NPC1 (0.41) MAPTALDH1A1HTTSMN1; SMN2LMNA
SCHEMBL17089944 0.81 ALDH1A1 (0.42) ACHEBACE1NPY5RPGRMAPT
SCHEMBL13565600 0.81 ALDH1A1 (0.42) ACHEBACE1NPY5RPGRMAPT
SCHEMBL10114238 0.81 SMN1; SMN2 (0.56) NPY5RMAPTHTTSMN1; SMN2RECQL
SCHEMBL13565429 0.80 BRD4 (0.41) NPY5RMAPTALDH1A1HTTLMNA
SCHEMBL17090178 0.80 CRHR1 (0.41) NPY5RCNR2EPHX2
SCHEMBL13565534 0.80 MAPT (0.41) MAPTALDH1A1SMN1; SMN2LMNACNR1
SCHEMBL13566025 0.80 CRHR1 (0.41) NPY5RCNR2EPHX2
SCHEMBL13565523 0.79 LMNA (0.38) MAPTALDH1A1SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed
US-8299265-B2 Amine derivatives having NPY Y5 receptor antagonistic activity and the uses thereof SHIONOGI & CO., LTD. (JP) 2012-10-30 US disclosed