SCHEMBL13565872

SCHEMBL13565872

CC(C)S(=O)(=O)NC1CCC(CNc2ccc(Nc3ccccc3)cc2)CC1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 2/20 0.41
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41
GRIA4 P48058 2/20 0.40
NPY5R Q15761 7/20 0.40
ALDH1A1 P00352 1/20 0.40
ALDH3A1 P30838 1/20 0.40
CARM1 Q86X55 1/20 0.40
PRMT6 Q96LA8 1/20 0.40
GRIA2 P42262 3/20 0.39
GBA1 P04062 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13565136 0.95 CRHR1 (0.44) CRHR1GRIA4NPY5RCARM1PRMT6
SCHEMBL17090375 0.95 CRHR1 (0.44) CRHR1GRIA4NPY5RCARM1PRMT6
SCHEMBL13439168 0.90 GRIA2 (0.44) CRHR1CNR1CNR2GRIA4NPY5R
SCHEMBL13565446 0.90 GRIA2 (0.44) CRHR1CNR1CNR2GRIA4NPY5R
SCHEMBL11941022 0.90 GRIA2 (0.44) CRHR1CNR1CNR2GRIA4NPY5R
SCHEMBL17090015 0.87 CRHR1 (0.47) CRHR1CNR1CNR2GRIA4NPY5R
SCHEMBL11935090 0.87 ACHE (0.41) CRHR1CNR1CNR2GRIA4NPY5R
SCHEMBL13564877 0.87 CRHR1 (0.47) CRHR1CNR1CNR2GRIA4NPY5R
SCHEMBL17090122 0.86 ALDH1A1 (0.42) CRHR1GRIA4NPY5RALDH1A1CARM1
SCHEMBL13113858 0.86 ALDH1A1 (0.42) CRHR1GRIA4NPY5RALDH1A1CARM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed
US-8299265-B2 Amine derivatives having NPY Y5 receptor antagonistic activity and the uses thereof SHIONOGI & CO., LTD. (JP) 2012-10-30 US disclosed