SCHEMBL13570548

SCHEMBL13570548

CC(C)Nc1cc(C(N)=O)ccc1Cl

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 1/20 0.54
ALDH1A1 P00352 2/20 0.47
MAPT P10636 1/20 0.47
KDM4E B2RXH2 1/20 0.47
HPGD P15428 2/20 0.46
BCAT2 O15382 1/20 0.46
LMNA P02545 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
MAPK14 Q16539 1/20 0.44
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
SLC6A3 Q01959 1/20 0.43
HDAC1 Q13547 3/20 0.42
HDAC8 Q9BY41 3/20 0.42
HDAC6 Q9UBN7 3/20 0.42
PARP1 P09874 1/20 0.41
HCAR3 P49019 1/20 0.40
F10 P00742 1/20 0.40
NPC1 O15118 1/20 0.40
ALOX12 P18054 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13736515 0.93 KDM4E (0.58) TOP2AALDH1A1MAPTKDM4EHPGD
SCHEMBL2104747 0.87 TOP2A (0.54) TOP2AALDH1A1KDM4EHPGDBCAT2
SCHEMBL28569255 0.75 TOP2A (0.50) TOP2AALDH1A1KDM4ELMNAMAPK14
SCHEMBL6114022 0.75 ALOX12 (0.50) ALDH1A1MAPTBCAT2LMNAHDAC1
SCHEMBL28623470 0.75 ALDH1A1 (0.49) ALDH1A1MAPTBCAT2MAPK14SLC6A2
SCHEMBL12125516 0.74 PARP1 (0.44) ALDH1A1MAPTKDM4EHPGDBCAT2
SCHEMBL7527111 0.73 KMT2A (0.53) ALDH1A1MAPTKDM4EHPGDBCAT2
SCHEMBL2105803 0.73 TOP2A (0.45) TOP2AMAPK14HCAR3
SCHEMBL4305366 0.73 CYP3A4 (0.46) ALDH1A1MAPTKDM4EHPGDLMNA
SCHEMBL8359924 0.72 RAPGEF4 (0.47) ALDH1A1MAPTHPGDLMNACA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012152983-A1 PHENYL- SULFONYL DERIVATIVES AS MEDIATORS OF TRPA1 RECEPTOR ACTIVITY FOR THE TREATMENT OF PAIN ORION CORPORATION (FI) 2012-11-15 WO disclosed
EP-2520566-A1 New Pharmaceutical Compounds Orion Corporation (FI) 2012-11-07 EP disclosed