SCHEMBL13577809

SCHEMBL13577809

Clc1ccc2cc(-c3ccc(N4CCNCC4)nc3)[nH]c2c1

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 1/20 0.52
HTR3B O95264 1/20 0.52
HTR3A P46098 1/20 0.52
HTR3D Q70Z44 1/20 0.52
HTR3C Q8WXA8 1/20 0.52
MGLL Q99685 3/20 0.46
FAAH O00519 1/20 0.45
MAP3K11 Q16584 1/20 0.44
CNR2 P34972 4/20 0.44
TNKS O95271 1/20 0.43
TLR9 Q9NR96 1/20 0.43
TLR8 Q9NR97 1/20 0.43
TLR7 Q9NYK1 1/20 0.43
DGAT1 O75907 4/20 0.42
KCNH2 Q12809 3/20 0.42
ADORA2A P29274 1/20 0.42
RET P07949 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1483676 0.87 TNKS (0.58) HTR3AMGLLTNKSTLR9TLR8
SCHEMBL1687841 0.78 HTR3E (0.54) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL12911533 0.78 GPR119 (0.58) HTR3EHTR3BHTR3AHTR3DHTR3C
Hydrochloric Acid SCHEMBL940785 0.76 GPR119 (0.56) HTR3EHTR3BHTR3AHTR3DHTR3C
Hydrochloric Acid SCHEMBL6786143 0.76 GPR119 (0.56) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL31195875 0.76 MGLL (0.48) MGLLCNR2TNKSTLR9TLR8
SCHEMBL1483695 0.75 KDM4E (0.40) MGLLRET
SCHEMBL1422658 0.75 PIM1 (0.40) MGLLCNR2
SCHEMBL194226 0.74 HTR3A (0.57) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL1483705 0.74 CNR1 (0.54) RET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009155024-A1 NOVEL SUBSTITUTED INDOLES MERCK & CO., INC. (US) 2009-12-23 WO disclosed