SCHEMBL13587

SCHEMBL13587

C=C1N=c2[nH]c(-c3ccc(F)cc3)cc2=CN1C1CCN(CCCCN)C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 2/20 0.35
HTR2A P28223 2/20 0.35
HRH4 Q9H3N8 3/20 0.34
CCNT1 O60563 2/20 0.32
CDK9 P50750 2/20 0.32
CHRM2 P08172 5/20 0.32
CHRM1 P11229 5/20 0.32
CHRM3 P20309 4/20 0.32
CHRNA3 P32297 1/20 0.30
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30
SLC22A2 O15244 1/20 0.30
MLNR O43193 1/20 0.30
CACNA1G O43497 1/20 0.30
CACNA1F O60840 1/20 0.30
GMNN O75496 1/20 0.30
USP2 O75604 1/20 0.30
USP1 O94782 1/20 0.30
KCNK2 O95069 1/20 0.30
CACNA1H O95180 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12061562 0.70 KIT (0.39) HRH4CHRM2CHRM1CHRM3CHRNA3
SCHEMBL14058 0.70 KIT (0.38) HRH4CHRM2CHRM1CHRM3CHRNA3
SCHEMBL3595429 0.56 DRD2 (0.59) HTR2AMEN1TP53CYP1A2CYP3A4
SCHEMBL11830521 0.56 SIGMAR1 (0.64) MEN1DRD2MAPK1KMT2A
SCHEMBL6972033 0.55 SCN5A (0.41) HTR2ACCNT1CDK9CHRM1CYP2D6
SCHEMBL228454 0.55 HTR2A (0.70) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL10978992 0.55
SCHEMBL855029 0.55 GNAI3 (0.40) CHRM3SLC6A4SMN1; SMN2HRH3
SCHEMBL855030 0.55 GNAI3 (0.40) CHRM3SLC6A4SMN1; SMN2HRH3
SCHEMBL856513 0.55 GNAI3 (0.40) CHRM3SLC6A4SMN1; SMN2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011047319-A2 ANTIMICROBIAL COMPOUNDS AND METHODS OF MAKING AND USING THE SAME RIB-X PHARMACEUTICALS, INC. (US) 2011-04-21 WO disclosed