SCHEMBL13600042

SCHEMBL13600042

Cc1nn(-c2ccc(C(F)(F)F)nc2)c(C)c1C=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.39
LMNA P02545 3/20 0.36
ALDH1A1 P00352 2/20 0.36
ALOX15 P16050 2/20 0.36
PTGS2 P35354 7/20 0.36
CYP2C9 P11712 2/20 0.36
TRPV4 Q9HBA0 1/20 0.36
PDPK1 O15530 2/20 0.35
PTGS1 P23219 2/20 0.35
PTGES O14684 1/20 0.35
HDAC3 O15379 1/20 0.35
CA12 O43570 1/20 0.35
PDE5A O76074 1/20 0.35
ABCB11 O95342 1/20 0.35
MT-CO2 P00403 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA3 P07451 1/20 0.35
CYP3A4 P08684 1/20 0.35
ALOX5 P09917 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5904596 0.80 BRAF (0.43) HTTLMNAALOX15PTGS2CYP2C9
SCHEMBL13600093 0.77 HTT (0.35) HTTLMNAALDH1A1ALOX15PTGS2
SCHEMBL27950463 0.75 LMNA (0.50) HTTLMNAALOX15PTGS2CYP2C9
SCHEMBL27875396 0.75 ALDH1A1 (0.49) HTTLMNAALDH1A1ALOX15MAPT
SCHEMBL24554045 0.73 KMT2A (0.55) HTTLMNAALDH1A1CYP3A4MAPT
SCHEMBL4239043 0.72 NPC1 (0.49) HTTLMNAALDH1A1ALOX15PTGS2
SCHEMBL13739457 0.72 MAPT (0.51) HTTLMNAALDH1A1ALOX15PTGS2
SCHEMBL1779819 0.71 HTT (0.64) HTTLMNAALDH1A1ALOX15MAPT
SCHEMBL28807415 0.71 CYP1A2 (0.55) HTTLMNAALDH1A1ALOX15CA1
SCHEMBL3321050 0.70 HTT (0.47) HTTLMNAALDH1A1ALOX15MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7625905-B2 Octahydro-pyrrolo[3,4-c]pyrrole CCR5 receptor antagonists ROCHE PALO ALTO LLC (US) 2009-12-01 US disclosed
US-20080103125-A1 Heterocylic antiviral compounds ROCHE PALO ALTO LLC 2008-05-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080103125-A1 Heterocylic antiviral compounds CCR5, ACKR3, CXCR3 HTT 2169/4885LMNA 4587/4885ALDH1A1 1201/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.