SCHEMBL13607802

SCHEMBL13607802

Brc1cnc2[nH]c(Cc3ccc4c(c3)OCO4)nc2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
HSD17B10 Q99714 2/20 0.44
MEN1 O00255 1/20 0.41
NPC1 O15118 1/20 0.41
LMNA P02545 1/20 0.41
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.41
MAPK1 P28482 3/20 0.41
FGFR1 P11362 1/20 0.40
FGFR2 P21802 1/20 0.40
TP53 P04637 1/20 0.40
MAPT P10636 1/20 0.40
L3MBTL1 Q9Y468 3/20 0.39
KDM4E B2RXH2 1/20 0.39
POLB P06746 1/20 0.39
APOBEC3A P31941 1/20 0.39
ESR2 Q92731 1/20 0.39
APOBEC3G Q9HC16 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
ADORA2A P29274 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4053745 0.81 ALDH1A1 (0.51) ALDH1A1HSD17B10MEN1NPC1LMNA
SCHEMBL13608086 0.79 PTPN7 (0.44) ALDH1A1HSD17B10MEN1NPC1LMNA
SCHEMBL13607799 0.78 CDK5 (0.48) ALDH1A1NPC1LMNARAB9AKMT2A
SCHEMBL13607804 0.78 LMNA (0.42) MEN1NPC1LMNARAB9AKMT2A
SCHEMBL13607793 0.78 RNASEH1 (0.43) ALDH1A1HSD17B10LMNAKMT2AMAPK1
SCHEMBL13607784 0.77 MAPT (0.40) MEN1NPC1LMNARAB9AKMT2A
SCHEMBL13607786 0.77 HPGD (0.44) ALDH1A1MEN1NPC1LMNARAB9A
SCHEMBL13607995 0.77 HPGD (0.45) ALDH1A1HSD17B10MEN1NPC1LMNA
SCHEMBL13607779 0.77 GAA (0.50) ALDH1A1NPC1LMNARAB9AKMT2A
SCHEMBL13607764 0.77 PARP1 (0.51) ALDH1A1HSD17B10MEN1LMNARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7622479-B2 Bicyclic derivative, its production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-24 US disclosed
US-7622479-B2 Bicyclic derivative, its production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-24 US disclosed