SCHEMBL13611375

SCHEMBL13611375

Cc1nc(Cc2ccc(-c3ccncc3)cc2)c[nH]1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 15/20 0.43
CYP11B1 P15538 12/20 0.43
CYP11B2 P19099 12/20 0.43
CYP3A4 P08684 7/20 0.42
CYP19A1 P11511 6/20 0.42
LMNA P02545 2/20 0.38
MAPT P10636 2/20 0.38
NPC1 O15118 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TP53 P04637 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KDM4E B2RXH2 1/20 0.37
CCNC P24863 1/20 0.35
CDK8 P49336 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11961681 0.81 CYP17A1 (0.41) CYP17A1CYP11B1CYP11B2CYP3A4CYP19A1
SCHEMBL10795179 0.81 ALDH1A1 (0.46) MAPTNPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL5037643 0.81 CYP17A1 (0.50) CYP17A1CYP11B1CYP11B2CYP3A4CYP19A1
SCHEMBL3840210 0.78 HSP90AB1 (0.45) LMNAMAPTNPC1TP53RAB9A
SCHEMBL13611413 0.78 HRH3 (0.42) LMNAMAPTNPC1ALDH1A1RAB9A
SCHEMBL16020932 0.78 MAPT (0.38) LMNAMAPTALDH1A1TP53SMN1; SMN2
SCHEMBL82538 0.78 TAAR1 (0.43) NPC1ALDH1A1RAB9ASMN1; SMN2
Water SCHEMBL10981448 0.76 TAAR1 (0.42) NPC1ALDH1A1RAB9ASMN1; SMN2KDM4E
SCHEMBL13611378 0.75 LTA4H (0.46) LMNAMAPTNPC1ALDH1A1RAB9A
Fluoride SCHEMBL28059937 0.75 TAAR1 (0.41) NPC1ALDH1A1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7625921-B2 Modulators of the glucocorticoid receptor, AP-1, and/or NF-κB activity and use thereof BRISTOL-MYERS SQUIBB COMPANY (US) 2009-12-01 US disclosed