SCHEMBL13616949

SCHEMBL13616949

Nc1ncsc1-c1cc(F)cc(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 3/20 0.44
ARNT P27540 4/20 0.36
EPAS1 Q99814 4/20 0.36
TDO2 P48775 1/20 0.33
DPP4 P27487 1/20 0.32
EPHB4 P54760 1/20 0.31
XPO1 O14980 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
THPO P40225 1/20 0.31
LMNA P02545 1/20 0.30
PMP22 Q01453 1/20 0.30
BRD4 O60885 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13616848 0.88 MAP4K4 (0.38) MAP4K4CYP1A2CYP3A4THPOLMNA
SCHEMBL13398555 0.75 KDM4E (0.54) MAP4K4ARNTEPAS1XPO1CYP1A2
SCHEMBL13616809 0.75 DHFR (0.47) MAP4K4TDO2DPP4
SCHEMBL13616873 0.70 CLK1 (0.37) MAP4K4DPP4EPHB4CYP3A4LMNA
SCHEMBL13398582 0.68 XPO1 (0.45) XPO1CYP1A2CYP3A4THPOLMNA
SCHEMBL13616861 0.62 PIM1 (0.40) EPHB4
SCHEMBL1231814 0.62 HSP90AA1 (0.36)
SCHEMBL17667859 0.61 ADORA2A (0.51)
SCHEMBL13616945 0.61 ADORA2A (0.48) CYP1A2CYP3A4BRD4
SCHEMBL10432894 0.61 KDM4E (0.35) CYP1A2CYP3A4THPOLMNAPMP22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2119716-A1 AZA-BRIDGED-RING COMPOUND Astellas Pharma Inc. (JP) 2009-11-18 EP disclosed