SCHEMBL13616848

SCHEMBL13616848

Nc1ncsc1-c1cc(F)cc(F)c1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 4/20 0.38
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
THPO P40225 1/20 0.34
LMNA P02545 1/20 0.33
PMP22 Q01453 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
PI4KA P42356 1/20 0.31
PI4K2B Q8TCG2 1/20 0.31
PI4K2A Q9BTU6 1/20 0.31
PI4KB Q9UBF8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13616949 0.88 MAP4K4 (0.44) MAP4K4CYP1A2CYP3A4THPOLMNA
SCHEMBL10432894 0.71 KDM4E (0.35) CYP1A2CYP3A4THPOLMNAPMP22
SCHEMBL9586083 0.71 KDM4E (0.62) CYP1A2CYP3A4THPOLMNAPMP22
SCHEMBL13616945 0.67 ADORA2A (0.48) ADORA2AADORA1CYP1A2CYP3A4
SCHEMBL13616808 0.67 ALDH1A1 (0.46) MAP4K4ADORA2AADORA1MEN1KMT2A
SCHEMBL12631776 0.67 HSD17B1 (0.49) MAP4K4ADORA1CYP3A4
SCHEMBL13616873 0.66 CLK1 (0.37) MAP4K4CYP3A4LMNAKDM4EMEN1
SCHEMBL13616805 0.65 MPL (0.47) MAP4K4ADORA2AADORA1KDM4E
SCHEMBL9586019 0.65 CYP1A2 (0.78) ADORA2ACYP1A2CYP3A4THPOLMNA
SCHEMBL1231814 0.64 HSP90AA1 (0.36) PI4KAPI4K2BPI4K2API4KB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2119716-A1 AZA-BRIDGED-RING COMPOUND Astellas Pharma Inc. (JP) 2009-11-18 EP disclosed