SCHEMBL13616945

SCHEMBL13616945

Nc1ncsc1-c1cccc(C(F)(F)F)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.48
ADORA1 P30542 2/20 0.48
IKBKB O14920 1/20 0.47
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
BRD4 O60885 1/20 0.43
RORB Q92753 2/20 0.43
RORC P51449 1/20 0.43
SCN2A Q99250 2/20 0.43
HRH1 P35367 1/20 0.43
HRH4 Q9H3N8 1/20 0.43
XDH P47989 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
PIK3CD O00329 1/20 0.41
PIK3CA P42336 1/20 0.41
PIK3CG P48736 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL984768 0.77 KDM4E (0.63) RORBRORCXDHCYP1A2CYP3A4
SCHEMBL13616808 0.76 ALDH1A1 (0.46) ADORA2AADORA1XDHPIK3CDPIK3CA
SCHEMBL12631776 0.76 HSD17B1 (0.49) ADORA1CYP3A4CYP2C9PIK3CDPIK3CA
SCHEMBL27803417 0.76 RORB (0.47) RORBRORCXDHCYP2C19ALDH1A1
SCHEMBL13616783 0.74 KDM4E (0.53) ADORA2AADORA1CYP1A2CYP3A4CYP2D6
SCHEMBL27803418 0.74 ALDH1A1 (0.46) RORBRORCALDH1A1
SCHEMBL982262 0.73 RORB (0.50) MAPK1RORBRORCCYP1A2CYP3A4
SCHEMBL28182113 0.73 TGFBR1 (0.51) ADORA2AADORA1RORBRORCSCN2A
SCHEMBL27732975 0.72 LTA4H (0.51) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL29678302 0.71 TSHR (0.58) TSHRMAPK1SCN2AALDH1A1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2119716-A1 AZA-BRIDGED-RING COMPOUND Astellas Pharma Inc. (JP) 2009-11-18 EP disclosed