SCHEMBL13618249

SCHEMBL13618249

CCCCCCCCOc1c(C)cc(C=O)cc1Br

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
THRA P10827 5/20 0.49
THRB P10828 5/20 0.49
S1PR2 O95136 7/20 0.43
S1PR1 P21453 7/20 0.43
S1PR3 Q99500 6/20 0.43
LPAR2 Q9HBW0 6/20 0.43
ALDH1A1 P00352 5/20 0.42
POLB P06746 2/20 0.42
KDM4E B2RXH2 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MAPK1 P28482 1/20 0.40
SRC P12931 1/20 0.40
LMNA P02545 1/20 0.39
S1PR4 O95977 2/20 0.39
S1PR5 Q9H228 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3903040 0.91 THRA (0.57) THRATHRBS1PR2S1PR1S1PR3
SCHEMBL8035224 0.89 THRA (0.51) THRATHRBS1PR2S1PR1S1PR3
SCHEMBL15498120 0.84 THRB (0.44) THRATHRBS1PR2S1PR1S1PR3
SCHEMBL3906365 0.83 ALDH1A1 (0.60) THRATHRBS1PR2S1PR1S1PR3
SCHEMBL14195848 0.83 ALDH1A1 (0.60) THRATHRBS1PR2S1PR1S1PR3
SCHEMBL14195849 0.83 ALDH1A1 (0.60) THRATHRBS1PR2S1PR1S1PR3
SCHEMBL14195841 0.83 ALDH1A1 (0.62) THRATHRBS1PR2S1PR1S1PR3
SCHEMBL14195854 0.83 ALDH1A1 (0.60) THRATHRBS1PR2S1PR1S1PR3
SCHEMBL14195852 0.83 ALDH1A1 (0.60) THRATHRBS1PR2S1PR1S1PR3
SCHEMBL9360147 0.83 ALDH1A1 (0.60) THRATHRBS1PR2S1PR1S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575964-B1 N-(BENZYL)AMINOALKYL CARBOXYLATE, PHOSPHINATES, PHOSPHONATES AND TETRAZOLES AS EDG RECEPTOR AGONISTS MERCK & CO INC (US) 2009-11-11 EP disclosed