SCHEMBL13619117

SCHEMBL13619117

CNS(=O)(=O)c1ccc(CC(C)C)c(C(=O)O)c1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.41
POLB P06746 3/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
KDM4E B2RXH2 2/20 0.40
BRAF P15056 1/20 0.39
TNNI3K Q59H18 1/20 0.39
ALDH1A1 P00352 1/20 0.39
ALDH3A1 P30838 1/20 0.39
NQO2 P16083 1/20 0.39
MTNR1A P48039 1/20 0.39
MAPK1 P28482 1/20 0.38
ATM Q13315 1/20 0.38
GAA P10253 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20033605 0.79 MAPK14 (0.36) LMNAPOLBMEN1KMT2ABRAF
SCHEMBL12338356 0.78 LMNA (0.42) LMNAL3MBTL1BRAFTNNI3KALDH1A1
SCHEMBL4420113 0.77 S1PR3 (0.47) LMNAKDM4EMAPK1
SCHEMBL19119211 0.75 POLB (0.59) LMNAPOLBL3MBTL1MEN1KMT2A
SCHEMBL2825786 0.75 ALDH1A1 (0.62) LMNAPOLBL3MBTL1MEN1KMT2A
SCHEMBL4901604 0.74 CA2 (0.50) LMNAPOLBL3MBTL1MEN1KMT2A
SCHEMBL3874483 0.74 MAPK1 (0.46) LMNAPOLBL3MBTL1MEN1KMT2A
SCHEMBL12225751 0.74 HSD17B10 (0.54) LMNAPOLBL3MBTL1MEN1KMT2A
SCHEMBL13543494 0.74 CYP3A4 (0.52) LMNAPOLBL3MBTL1MEN1KMT2A
SCHEMBL4844487 0.74 KMT2A (0.50) LMNAPOLBL3MBTL1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1848694-B1 HETEROCYCLIC SUBSTITUTED PHENYL METHANONES AS INHIBITORS OF THE GLYCINE TRANSPORTER 1 HOFFMANN LA ROCHE (CH) 2009-11-25 EP disclosed