SCHEMBL13625938

SCHEMBL13625938

CCc1nc(C)n(-c2ccccc2)c(=O)c1CC1=CC=C(c2ccccc2C#N)CC1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.34
ALOX15 P16050 1/20 0.34
ATM Q13315 1/20 0.34
HSD17B10 Q99714 1/20 0.34
KDM5A P29375 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TP53 P04637 2/20 0.33
TDP2 O95551 1/20 0.32
KDM4E B2RXH2 1/20 0.32
GAA P10253 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
FPR1 P21462 1/20 0.32
CYP2C19 P33261 1/20 0.32
LMNA P02545 2/20 0.31
HCRTR1 O43613 1/20 0.31
NOS2 P35228 1/20 0.31
DPP4 P27487 2/20 0.31
F10 P00742 1/20 0.31
GRIA1 P42261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1894719 0.80 KDM4E (0.40) ALDH1A1ALOX15ATMHSD17B10KDM4E
SCHEMBL13625909 0.76 ACHE (0.34)
SCHEMBL27771409 0.74 CYP19A1 (0.41) ALDH1A1KDM5ANPSR1KDM4EGAA
SCHEMBL1893086 0.73 PPARG (0.45)
SCHEMBL27792506 0.72 PPARG (0.36) ALDH1A1KDM5AKDM4EGAACYP2D6
SCHEMBL2871115 0.72 ACHE (0.45)
SCHEMBL13626516 0.70 AGTR1 (0.33) ALDH1A1KDM4E
SCHEMBL12348734 0.70 PPARG (0.40) ALDH1A1KDM5AKDM4EGAACYP2D6
SCHEMBL1892338 0.70 APLNR (0.36) CYP2C19MAPT
SCHEMBL4013362 0.69 MAPK1 (0.37) ALDH1A1ALOX15ATMHSD17B10TDP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009133970-A1 CRYSTALLINE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-05 WO disclosed