SCHEMBL13626823

SCHEMBL13626823

CCc1sc(C(=O)Nc2c(C)ccc(-c3cc(Nc4ccc(C5CCN(C)CC5)nn4)c(=O)n(C)c3)c2Cl)cc1C(C)C

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCND1 P24385 2/20 0.40
CDK6 Q00534 1/20 0.40
BTK Q06187 16/20 0.38
CDK4 P11802 1/20 0.34
RAF1 P04049 1/20 0.33
BRAF P15056 1/20 0.33
CLK2 P49760 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13626372 0.89 CCND1 (0.46) CCND1CDK6BTKCDK4
SCHEMBL13626127 0.88 CCND1 (0.43) CCND1CDK6BTKCDK4
SCHEMBL13626138 0.85 BTK (0.51) BTK
SCHEMBL1422433 0.84 BTK (0.39) CCND1CDK6BTKRAF1BRAF
SCHEMBL13626377 0.84 CDK6 (0.45) CCND1CDK6BTKCDK4CLK2
SCHEMBL13626378 0.83 CCND1 (0.47) CCND1CDK6BTKCDK4
SCHEMBL13626188 0.82 CDK6 (0.45) CCND1CDK6BTKCDK4
SCHEMBL13626142 0.74 BTK (0.54) BTK
SCHEMBL1422829 0.73 CCND1 (0.40) CCND1CDK6BTK
SCHEMBL1422539 0.72 BTK (0.39) CCND1CDK6BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009137596-A1 SUBSTITUTED AMIDES, METHOD OF MAKING, AND USE AS BTK INHIBITORS CGI PHARMACEUTICALS, INC. (US) 2009-11-12 WO disclosed