SCHEMBL13627398

SCHEMBL13627398

NC(=O)c1cccc2ccc(-c3cccc(C(F)(F)F)c3)nc12

nearest known ligand 0.67

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 9/20 0.67
KMO O15229 2/20 0.50
CTSS P25774 1/20 0.48
JAK2 O60674 2/20 0.46
KDM4E B2RXH2 1/20 0.46
KDM1A O60341 2/20 0.45
XDH P47989 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1035363 0.88 KMO (0.57) PARP1KMOCTSSKDM4EKDM1A
SCHEMBL13854087 0.82 CTSS (0.58) KMOCTSSKDM4EKDM1AXDH
SCHEMBL1034065 0.81 RXFP1 (0.53) PARP1
SCHEMBL6442515 0.81 PARP1 (1.00) PARP1KDM4E
SCHEMBL31061508 0.81 PARP1 (1.00) PARP1KDM4E
SCHEMBL1034305 0.80 KMO (0.49) PARP1KMO
SCHEMBL17772322 0.80 KMO (0.44) PARP1KMOCTSSKDM4EKDM1A
SCHEMBL1032856 0.80 KDM1A (0.50) PARP1KMOCTSSKDM4EKDM1A
SCHEMBL1034072 0.79 JAK2 (0.51) KMOJAK2
SCHEMBL27830698 0.79 ALDH1A1 (0.54) PARP1KMOKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009134973-A1 QUENOLINES AND RELATED ANALOGS AS SIRTUIN MODULATORS SIRTRIS PHARMACEUTICALS, INC. (US) 2009-11-05 WO disclosed