SCHEMBL13627977

SCHEMBL13627977

COc1cc(CN2C(=O)/C(=N\O)c3cc(F)ccc32)cc(OC)c1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.43
CHRM5 P08912 4/20 0.43
ALDH1A1 P00352 4/20 0.42
ALDH3A1 P30838 4/20 0.42
PARK7 Q99497 2/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
UCHL3 P15374 3/20 0.39
UCHL1 P09936 2/20 0.39
ACE P12821 1/20 0.39
WDR5 P61964 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13627970 0.91 CHRM5 (0.53) TRPA1CHRM5ALDH1A1ALDH3A1CA12
SCHEMBL13627966 0.86 UCHL3 (0.52) CHRM5ALDH1A1ALDH3A1CA12CA1
SCHEMBL13628006 0.84 CHRM5 (0.63) CHRM5
SCHEMBL13627958 0.84 ALDH1A1 (0.52) CHRM5ALDH1A1ALDH3A1PARK7ACE
SCHEMBL13627937 0.84 CHRM5 (0.55) TRPA1CHRM5ALDH1A1ALDH3A1PARK7
SCHEMBL13628017 0.84 CA12 (0.47) CA12CA1CA2CA9
SCHEMBL13627940 0.82 CHRM5 (0.51) TRPA1CHRM5ALDH1A1ALDH3A1PARK7
SCHEMBL13628069 0.82 CHRM5 (0.47) CHRM5ALDH1A1PARK7CA12CA1
SCHEMBL13627936 0.82 TRPA1 (0.62) TRPA1CHRM5ALDH1A1ALDH3A1PARK7
SCHEMBL13627946 0.81 UBE2N (0.56) TRPA1CHRM5ALDH1A1ALDH3A1PARK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612065-B2 Inhibitors of c-JUN N-terminal kinases (JNK) VERTEX PHARMACEUTICALS INCORPORATED (US) 2009-11-03 US disclosed
US-7612065-B2 Inhibitors of c-JUN N-terminal kinases (JNK) VERTEX PHARMACEUTICALS INCORPORATED (US) 2009-11-03 US disclosed
US-20080033022-A1 Inhibitors of c-Jun N-terminal kinases (JNK) SALITURO FRANCESCO G 2008-02-07 US disclosed
US-20080033022-A1 Inhibitors of c-Jun N-terminal kinases (JNK) SALITURO FRANCESCO G 2008-02-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080033022-A1 Inhibitors of c-Jun N-terminal kinases (JNK) MAP3K1, JUN, MAP3K7 TRPA1 4561/4885CHRM5 4815/4885ALDH1A1 4310/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.